SCHEMBL5282876

SCHEMBL5282876

O=C1c2ccc(O)cc2CN1Cc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.49
HDAC4 P56524 2/20 0.49
HDAC6 Q9UBN7 2/20 0.49
GRM5 P41594 1/20 0.49
PARP1 P09874 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
PRMT5 O14744 1/20 0.46
WDR77 Q9BQA1 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
ACHE P22303 2/20 0.46
DHPS P49366 1/20 0.45
ADAM17 P78536 1/20 0.45
KDM4E B2RXH2 1/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
SIRT1 Q96EB6 1/20 0.44
PREP P48147 1/20 0.44
ESR1 P03372 1/20 0.43
ESR2 Q92731 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31409566 1.00 HDAC1 (0.49) HDAC1HDAC4HDAC6GRM5PARP1
SCHEMBL16850291 0.88 HDAC1 (0.58) HDAC1HDAC4HDAC6GRM5PARP1
SCHEMBL21768036 0.88 ERCC1 (0.47) HDAC1MEN1KMT2APRMT5WDR77
SCHEMBL2023150 0.87 GRM5 (0.50) HDAC1HDAC4HDAC6GRM5PARP1
SCHEMBL3054839 0.86 GRM5 (0.67) GRM5PRMT5WDR77ACHEDHPS
SCHEMBL31409495 0.86 PARP1 (0.50) PARP1KMT2APRMT5WDR77ACHE
SCHEMBL31409533 0.86 ADAM17 (0.57) MEN1KMT2AADAM17
SCHEMBL31409508 0.86 CYP19A1 (0.50) HDAC1HDAC4HDAC6MEN1KMT2A
SCHEMBL29438631 0.86 GRM5 (0.67) GRM5PRMT5WDR77ACHEDHPS
SCHEMBL31409506 0.84 DHPS (0.51) HDAC1HDAC4HDAC6MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007000337-A1 BICYCLIC DERIVATIVES AS P38 KINASE INHIBITORS PALAU PHARMA, S.A. (ES) 2007-01-04 WO disclosed