SCHEMBL5287809

SCHEMBL5287809

Cn1nc(-c2ccc(CNCCNC(=O)OC(C)(C)C)cc2)ccc1=O

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.44
CD274 Q9NZQ7 1/20 0.44
HRH3 Q9Y5N1 4/20 0.43
GLA P06280 1/20 0.40
TP53 P04637 3/20 0.40
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.39
PPARG P37231 1/20 0.39
PPARD Q03181 1/20 0.39
PPARA Q07869 1/20 0.39
MAPT P10636 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
GFER P55789 1/20 0.37
PHGDH O43175 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5324144 0.77 HRH3 (0.38) HRH3GLATP53KDM4EALDH1A1
SCHEMBL4415421 0.76 GAA (0.56) PDCD1CD274PPARACA1CA2
SCHEMBL21066539 0.75 PDCD1 (0.49) PDCD1CD274CA1CA2L3MBTL1
SCHEMBL4709745 0.75 PDCD1 (0.52) PDCD1CD274TP53MAPTSMN1; SMN2
SCHEMBL29904798 0.75 L3MBTL1 (0.48) KDM4EMAPTCA1CA2L3MBTL1
SCHEMBL6076877 0.74 HPGD (0.49) PDCD1CD274KDM4EALDH1A1CA1
SCHEMBL12310009 0.74 CA1 (0.47) PDCD1CD274CA1CA2L3MBTL1
SCHEMBL1724201 0.74 GAA (0.60) PDCD1CD274KDM4EALDH1A1SMN1; SMN2
SCHEMBL22452272 0.74 FPR3 (0.47) PDCD1CD274SMN1; SMN2CA1CA2
SCHEMBL5479565 0.74 CYP17A1 (0.50) PDCD1CD274ALDH1A1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007008144-A1 HETEROCYCLIC SULFONAMIDE DERIVATIVES AS INHIBITORS OF FACTOR XA ASTRAZENECA AB (SE) 2007-01-18 WO disclosed