SCHEMBL528806

SCHEMBL528806

CC(COC(N)=O)c1ccc(N=Nc2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 8/20 0.51
CYP1A2 P05177 3/20 0.51
PKM P14618 2/20 0.51
CYP2D6 P10635 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
MAPT P10636 9/20 0.46
RAB9A P51151 8/20 0.46
NPC1 O15118 5/20 0.46
ALDH1A1 P00352 5/20 0.46
MEN1 O00255 5/20 0.46
KMT2A Q03164 5/20 0.46
LMNA P02545 3/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
TDP1 Q9NUW8 1/20 0.46
CASP3 P42574 1/20 0.43
SENP8 Q96LD8 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
SENP6 Q9GZR1 1/20 0.43
HPGD P15428 2/20 0.42
TRPA1 O75762 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4589554 0.86 CYP1A2 (0.68) SMN1; SMN2CYP1A2PKMCYP2D6NPSR1
SCHEMBL28958757 0.86 CYP1A2 (0.68) SMN1; SMN2CYP1A2PKMCYP2D6NPSR1
SCHEMBL4590669 0.86 CYP1A2 (0.68) SMN1; SMN2CYP1A2PKMCYP2D6NPSR1
SCHEMBL528539 0.83 CYP1A2 (0.56) SMN1; SMN2CYP1A2PKMCYP2D6NPSR1
SCHEMBL20563823 0.83 CYP1A2 (0.56) SMN1; SMN2CYP1A2PKMCYP2D6NPSR1
SCHEMBL994448 0.77 MAPT (0.46) SMN1; SMN2CYP1A2PKMCYP2D6MAPT
SCHEMBL994450 0.77 MAPT (0.46) SMN1; SMN2CYP1A2PKMCYP2D6MAPT
SCHEMBL29213688 0.76 ALOX5 (0.47) SMN1; SMN2CYP1A2PKMCYP2D6NPSR1
SCHEMBL3468423 0.76 ALOX5 (0.47) SMN1; SMN2CYP1A2PKMCYP2D6NPSR1
Azobenzene SCHEMBL28244550 0.76 ALOX15 (0.56) SMN1; SMN2CYP1A2PKMCYP2D6NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 175 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4724418-A1 TRICINE AND CITRIC ACID-BASED CATIONIC LIPIDS Sanofi (FR) 2026-04-15 EP disclosed
WO-2025054361-A1 COMPLEMENT INHIBITION APELLIS PHARMACEUTICALS, INC. (US) 2025-03-13 WO disclosed
EP-4486336-A2 CB1 LIGAND CONJUGATED COMPOUNDS AND USES THEREOF Adarx Pharmaceuticals, Inc. (US) 2025-01-08 EP disclosed
WO-2025003759-A1 DIANHYDROHEXITOL BASED IONIZABLE LIPIDS FOR NUCLEIC ACID DELIVERY SANOFI (FR) 2025-01-02 WO disclosed
EP-4475837-A2 TRKB LIGAND CONJUGATED COMPOUNDS AND USES THEREOF Adarx Pharmaceuticals, Inc. (US) 2024-12-18 EP disclosed
WO-2024148274-A1 COMPLEMENT INHIBITION APELLIS PHARMACEUTICALS, INC. (US) 2024-07-11 WO disclosed
EP-4362933-A1 COMPLEMENT INHIBITION Apellis Pharmaceuticals, Inc. (US) 2024-05-08 EP disclosed
EP-4340859-A1 ANTIBODY DRUG CONJUGATES USING MATES TECHNOLOGY FOR DELIVERING CYTOTOXIC AGENTS Biohaven Therapeutics Ltd. (US) 2024-03-27 EP disclosed
EP-4323346-A1 GOOD\"BUFFER-BASED CATIONIC LIPIDS Translate Bio, Inc. (US) 2024-02-21 EP disclosed
EP-4288465-A1 ACTIVE AGENT-RELEASING HYALURONIC ACID VEHICLE Ariel Scientific Innovations Ltd. (IL) 2023-12-13 EP disclosed
WO-2011073967-A1 A BIOMATERIAL VYSERA BIOMEDICAL LIMITED (IE) 2011-06-23 WO disclosed
EP-2303897-A1 HIGH-VALENT PALLADIUM FLUORIDE COMPLEXES AND USES THEREOF President and Fellows of Harvard College (US) 2011-04-06 EP disclosed
WO-2011006088-A2 FLUORINE CONTAINING COMPOUNDS AND METHODS OF USE THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2011-01-13 WO disclosed
WO-2010059241-A2 TREATMENT OF AMYOTROPHIC LATERAL SCLEROSIS CAMBRIA PHARMACEUTICALS, INC. (US) 2010-05-27 WO disclosed
WO-2010011313-A2 LIGATION OF STAPLED POLYPEPTIDES PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2010-01-28 WO disclosed
WO-2009149347-A1 HIGH-VALENT PALLADIUM FLUORIDE COMPLEXES AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2009-12-10 WO disclosed
WO-2008124571-A2 ANTI-VIRAL COMPOUNDS, COMPOSITIONS AND METHODS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2008-10-16 WO disclosed
WO-2008028057-A2 SHIKIMIC ACID-DERIVED COMPOUNDS FOR INHIBITION AND DETECTION OF AURORA A-ASSOCIATED TUMORS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2008-03-06 WO disclosed
EP-0970066-A1 AMINOEPOXIDES FROM AMINOALDEHYDES AND IN-SITU FORMED HALOMETHYL ORGANOMETALLIC REAGENT G.D. SEARLE & CO. (US) 2000-01-12 EP disclosed
WO-1998029401-A1 AMINOEPOXIDES FROM AMINOALDEHYDES AND IN-SITU FORMED HALOMETHYL ORGANOMETALLIC REAGENT G.D. SEARLE & CO. (US) 1998-07-09 WO disclosed