SCHEMBL5289381

SCHEMBL5289381

Cc1ccc(CC(=O)Nc2ccc3ncn(C(CC(=O)O)c4ccccc4)c3c2)cc1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 4/20 0.44
ITGA4 P13612 4/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
KDM4E B2RXH2 1/20 0.44
TP53 P04637 1/20 0.44
MAPT P10636 1/20 0.44
NLRP3 Q96P20 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.42
NAMPT P43490 1/20 0.42
NOTUM Q6P988 2/20 0.42
KDR P35968 3/20 0.41
WNT3A P56704 1/20 0.41
FNTA P49354 1/20 0.41
FNTB P49356 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2294482 0.93 NAMPT (0.48) ITGB1ITGA4NPC1RAB9AKDM4E
SCHEMBL5305129 0.93 NPC1 (0.49) ITGB1ITGA4NPC1RAB9AKDM4E
SCHEMBL2298594 0.91 KMT2A (0.46) ITGB1ITGA4NPC1RAB9AKDM4E
SCHEMBL2295665 0.91 PSEN1 (0.45) ITGB1ITGA4NPC1RAB9AKDM4E
SCHEMBL2294562 0.91 MAPT (0.44) ITGB1ITGA4NPC1RAB9AKDM4E
SCHEMBL2292763 0.90 MAPT (0.50) RAB9AKDM4EMAPTNLRP3SMN1; SMN2
SCHEMBL5291502 0.88 BCHE (0.46) ITGB1ITGA4NPC1RAB9AKDM4E
SCHEMBL2294711 0.87 ALDH1A1 (0.47) KDM4EMAPTSMN1; SMN2NAMPTFNTA
SCHEMBL2299138 0.87 NOTUM (0.46) ITGB1ITGA4NPC1RAB9AMAPT
SCHEMBL2292564 0.87 NPC1 (0.51) NPC1RAB9AKDM4ETP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828144-A2 INTEGRIN ANTAGONISTS USEFUL AS ANTICANCER AGENTS OSI Pharmaceuticals, Inc. (US) 2007-09-05 EP claimed
WO-2006053342-A2 INTEGRIN ANTAGONISTS USEFUL AS ANTICANCER AGENTS OSI PHARMACEUTICALS, INC. (US) 2006-05-18 WO claimed