SCHEMBL5289451

SCHEMBL5289451

Cc1cc(I)cc([N+](=O)[O-])c1

nearest known ligand 0.71

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.71
HTT P42858 3/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
LMNA P02545 1/20 0.52
ACHE P22303 2/20 0.50
HSD17B10 Q99714 1/20 0.46
CYP19A1 P11511 1/20 0.44
ALDH1A1 P00352 4/20 0.42
GPR35 Q9HC97 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
CYP3A4 P08684 2/20 0.39
POLB P06746 1/20 0.39
GALR3 O60755 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1097495 0.84 TSHR (1.00) TSHRHTTMEN1KMT2ALMNA
SCHEMBL309438 0.84 CYP19A1 (0.62) TSHRHTTMEN1KMT2ALMNA
SCHEMBL222935 0.84 LMNA (0.56) TSHRHTTMEN1KMT2ALMNA
SCHEMBL635130 0.84 TSHR (0.90) TSHRHTTMEN1KMT2ALMNA
Ammonia Solution, Strong SCHEMBL27814867 0.75 TSHR (0.49) TSHRHTTMEN1KMT2ALMNA
SCHEMBL16955649 0.74 LMNA (0.47) TSHRHTTMEN1KMT2ALMNA
SCHEMBL220173 0.74 LMNA (0.47) TSHRHTTMEN1KMT2ALMNA
SCHEMBL1171962 0.74 LMNA (0.47) TSHRHTTMEN1KMT2ALMNA
SCHEMBL9452187 0.74 ALDH1A1 (0.50) TSHRHTTMEN1KMT2ALMNA
SCHEMBL29920469 0.74 LMNA (0.47) TSHRHTTMEN1KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017089800-A1 MICROBUBBLE-CHEMOTHERAPEUTIC AGENT COMPLEX FOR SONODYNAMIC THERAPY UNIVERSITY OF ULSTER (GB) 2017-06-01 WO disclosed
EP-2900645-A1 3-PHENYLISOXAZOLIN DERIVATIVES WITH HERBICIDAL ACTION Bayer CropScience AG (DE) 2015-08-05 EP disclosed
CN-102115452-A (E)-3-(3-substituted-5-methylphenyl)acrylonitrile and preparation method thereof TOPHARMAN SHANGHAI CO LTD 2011-07-06 CN disclosed
WO-2006129120-A9 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2007-03-22 WO disclosed
WO-2006129120-A2 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2006-12-07 WO disclosed
US-5270309-A Kynurenic acid derivatives useful in the treatment of neurodegenerative disorders MERCK SHARP & DOHME LIMITED (GB) 1993-12-14 US disclosed
EP-0303387-B1 KYNURENIC ACID DERIVATIVES USEFUL IN THE TREATMENT OF NEURODEGENERATIVE DISORDERS MERCK SHARP & DOHME LTD. (GB) 1993-04-21 EP disclosed
EP-0303387-A1 Kynurenic acid derivatives useful in the treatment of neurodegenerative disorders MERCK SHARP & DOHME LTD. (GB) 1989-02-15 EP disclosed