SCHEMBL5289989

SCHEMBL5289989

c1ccc(NCCC2CCCN2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 3/20 0.50
MAN1B1 Q9UKM7 1/20 0.48
POLB P06746 1/20 0.47
KMT2A Q03164 1/20 0.46
CHRNB4 P30926 2/20 0.43
CHRNA3 P32297 2/20 0.43
CHRNB2 P17787 2/20 0.43
CHRNA4 P43681 2/20 0.43
CHRNA1 P02708 1/20 0.43
CHRNG P07510 1/20 0.43
CHRNB1 P11230 1/20 0.43
CHRND Q07001 1/20 0.43
METAP2 P50579 1/20 0.43
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3329262 0.83 LTA4H (0.52) LTA4HPOLBCHRNB4CHRNA3CHRNB2
SCHEMBL1116568 0.83 LTA4H (0.52) LTA4HPOLBCHRNB4CHRNA3CHRNB2
SCHEMBL1116569 0.83 LTA4H (0.52) LTA4HPOLBCHRNB4CHRNA3CHRNB2
SCHEMBL11969843 0.82 LTA4H (0.42) LTA4HPOLBKMT2AMETAP2CYP1A2
SCHEMBL10891765 0.80 LTA4H (0.49) LTA4HCYP1A2CYP2D6CYP2C19SMN1; SMN2
SCHEMBL4374404 0.78 POLB (0.57) LTA4HPOLBKMT2ACYP1A2CYP2D6
SCHEMBL4381640 0.77 POLB (0.56) LTA4HPOLBKMT2ACYP1A2CYP2D6
SCHEMBL4654443 0.74 LTA4H (0.51) LTA4HPOLBCHRNB4CHRNA3CHRNB2
SCHEMBL1751545 0.74 LTA4H (0.51) LTA4HPOLBCHRNB4CHRNA3CHRNB2
SCHEMBL3289066 0.74 ACHE (0.52) ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863805-A1 PYRIMIDINE COMPOUNDS HAVING TIE2 (TEK) INHIBITORY ACTIVITY AstraZeneca AB (SE) 2007-12-12 EP disclosed
WO-2006082373-A1 PYRIMIDINE COMPOUNDS HAVING TIES (TEK) INHIBITORY ACTIVITY ASTRAZENECA AB (SE) 2006-08-10 WO disclosed