SCHEMBL529465

SCHEMBL529465

O=C(O)c1cnc2ccc(-c3ccncc3)cc2c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 1/20 0.63
CDK8 P49336 1/20 0.63
CLK2 P49760 1/20 0.63
CDK7 P50613 1/20 0.63
CDK9 P50750 1/20 0.63
CDK5 Q00535 1/20 0.63
ACVR1 Q04771 1/20 0.63
ROCK1 Q13464 1/20 0.63
DYRK1A Q13627 1/20 0.63
LRRK2 Q5S007 1/20 0.63
CLK4 Q9HAZ1 1/20 0.63
DYRK1B Q9Y463 1/20 0.63
MGAM O43451 1/20 0.55
PDGFRB P09619 7/20 0.49
PDGFRA P16234 7/20 0.49
EGFR P00533 1/20 0.49
IP6K1 Q92551 1/20 0.47
IP6K3 Q96PC2 1/20 0.47
IP6K2 Q9UHH9 1/20 0.47
BRAF P15056 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4398475 0.88 MGAM (0.68) MAP4K4CDK8CLK2CDK7CDK9
SCHEMBL529524 0.86 MGAM (0.57) MAP4K4CDK8CLK2CDK7CDK9
SCHEMBL1352698 0.84 MAP4K4 (0.58) MAP4K4CDK8CLK2CDK7CDK9
SCHEMBL10465639 0.80 MGAM (0.70) MGAMPDGFRBPDGFRANAPRT
SCHEMBL12504970 0.79 MGAM (0.56) MAP4K4CDK8CLK2CDK7CDK9
SCHEMBL3787407 0.79 MGAM (0.64) MGAMCSNK2A2CSNK2BNAPRT
SCHEMBL12132266 0.78 MGAM (0.51) MAP4K4CDK8CLK2CDK7CDK9
SCHEMBL528875 0.77 MGAM (0.54) MGAMPDGFRBPDGFRA
SCHEMBL28055368 0.76 MGAM (0.60) MAP4K4MGAMPDGFRBPDGFRAMKNK1
SCHEMBL61876 0.76 MGAM (0.64) MAP4K4CDK8CLK2CDK7CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597955-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-06-05 EP disclosed
WO-2012016082-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2012-02-02 WO disclosed