SCHEMBL5299057

SCHEMBL5299057

CCSc1nnc(C)c(O)n1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.38
ALDH1A1 P00352 2/20 0.37
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ABCB1 P08183 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
KDM4E B2RXH2 1/20 0.32
CYP1A2 P05177 1/20 0.32
CASP7 P55210 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14611721 0.84 ALDH1A1 (0.42) ALDH1A1HPGDHTTRAB9ASMN1; SMN2
SCHEMBL14611718 0.81 USP2 (0.43) ALDH1A1HPGDTSHRHTTRAB9A
SCHEMBL14611586 0.79 LMNA (0.41) ALDH1A1HPGDRAB9ASMN1; SMN2MEN1
SCHEMBL3236065 0.77 MAPT (0.45) ALDH1A1HPGDTSHRMAPK1RAB9A
SCHEMBL14611587 0.77 KDM1A (0.34) ALDH1A1HPGDRAB9ASMN1; SMN2KDM4E
SCHEMBL14611585 0.76 POLB (0.33) ALDH1A1RAB9AHSD17B10TDP1KDM4E
SCHEMBL14611713 0.76 MAPT (0.37) ALDH1A1HPGDMAPK1HTTSMN1; SMN2
SCHEMBL14611583 0.73 ALDH1A1 (0.53) HSP90AA1ALDH1A1HPGDTSHRMAPK1
SCHEMBL7020481 0.72 KMT2A (0.41) HSP90AA1ALDH1A1RAB9ASMN1; SMN2KDM4E
SCHEMBL5305067 0.72 PDPK1 (0.35) HSP90AA1ALDH1A1ABCB1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007017114-A1 NEW SUBSTITUTED AZATHYMIDINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF BACTERIAL INFECTIOUS DISEASES MERLION PHARMACEUTICALS SA (CH) 2007-02-15 WO claimed
WO-2007017114-A1 NEW SUBSTITUTED AZATHYMIDINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF BACTERIAL INFECTIOUS DISEASES MERLION PHARMACEUTICALS SA (CH) 2007-02-15 WO disclosed
WO-2007017114-A1 NEW SUBSTITUTED AZATHYMIDINE DERIVATIVES AND THEIR USE IN THE TREATMENT OF BACTERIAL INFECTIOUS DISEASES MERLION PHARMACEUTICALS SA (CH) 2007-02-15 WO disclosed