SCHEMBL5300690

SCHEMBL5300690

CCI.CCn1c(COCc2ccccc2)nc(C(C)C)c1Sc1cc(C#N)cc(C#N)c1

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.34
VCP P55072 1/20 0.34
MCL1 Q07820 1/20 0.32
MAOB P27338 1/20 0.32
GHSR Q92847 2/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
ACSS2 Q9NR19 1/20 0.32
TLR7 Q9NYK1 1/20 0.31
CYP19A1 P11511 1/20 0.31
HTR2C P28335 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4900234 0.97 TSHR (0.36) TSHRVCPMCL1MAOBGHSR
SCHEMBL4898932 0.85 VCP (0.36) TSHRVCPMCL1MAOBGHSR
SCHEMBL4899994 0.84 TSHR (0.37) TSHRVCPMAOBGHSRMAPT
SCHEMBL6966496 0.82 VCP (0.37) TSHRVCPTP53MAPTACSS2
SCHEMBL6960428 0.82 VCP (0.37) TSHRVCPACSS2
SCHEMBL5243251 0.82 HTR2C (0.32) TLR7HTR2C
SCHEMBL4901053 0.81 TSHR (0.37) TSHRMAOBGHSRACSS2HTR2C
SCHEMBL4902092 0.81 TSHR (0.35) TSHRMAOBGHSRACSS2HTR2C
SCHEMBL6960598 0.79 TDP1 (0.36) TSHRVCPTP53
SCHEMBL6957486 0.79 VCP (0.36) TSHRVCPTP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740550-A1 SULPHUR-LINKED IMIDAZOLE COMPOUNDS FOR THE TREAMENT OF HIV Pfizer Limited (GB) 2007-01-10 EP disclosed
WO-2005100322-A1 SULPHUR-LINKED IMIDAZOLE COMPOUNDS FOR THE TREAMENT OF HIV PFIZER LIMITED (GB) 2005-10-27 WO disclosed