SCHEMBL6966496

SCHEMBL6966496

CCn1c(COCc2ccccc2)nc(C(C)C)c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
VCP P55072 1/20 0.37
TDP1 Q9NUW8 1/20 0.35
TP53 P04637 2/20 0.33
DHODH Q02127 2/20 0.33
MAPT P10636 1/20 0.32
TACR1 P25103 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
SLC5A2 P31639 1/20 0.32
TSHR P16473 1/20 0.31
ACSS2 Q9NR19 1/20 0.31
ADAMTS5 Q9UNA0 2/20 0.31
MMP2 P08253 1/20 0.31
MMP13 P45452 1/20 0.31
ADAM17 P78536 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14439828 0.93 TDP1 (0.40) VCPTDP1TP53DHODHMAPT
SCHEMBL6960598 0.92 TDP1 (0.36) VCPTDP1TP53TACR1L3MBTL1
SCHEMBL14439841 0.91 VCP (0.36) VCPTDP1TP53DHODHMAPT
SCHEMBL14439829 0.91 VCP (0.36) VCPTDP1TP53DHODHMAPT
SCHEMBL6965896 0.91 VCP (0.36) VCPTDP1TP53DHODHMAPT
SCHEMBL6972304 0.90 HSP90B1 (0.37) VCPTDP1DHODHMAPTSMN1; SMN2
SCHEMBL6974348 0.89 GSK3B (0.34) VCPTDP1TACR1L3MBTL1
SCHEMBL6974229 0.89 MAPT (0.34) TP53DHODHMAPTNPC1RAB9A
SCHEMBL6973959 0.89 VCP (0.35) VCPTDP1TP53DHODHMAPT
SCHEMBL14439830 0.89 TP53 (0.39) VCPTDP1TP53DHODHMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed