SCHEMBL5301651

SCHEMBL5301651

O=C(O)CC(c1ccccc1)n1cnc2ccc(NC(=O)C3CC4C=CC3C4)cc21

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.39
ALDH1A1 P00352 8/20 0.34
KDM4E B2RXH2 3/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2C19 P33261 2/20 0.34
MAPT P10636 2/20 0.34
HPGD P15428 1/20 0.34
LMNA P02545 3/20 0.33
RAB9A P51151 2/20 0.33
NPC1 O15118 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NOTUM Q6P988 2/20 0.33
MAPK1 P28482 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5288809 0.93 RAB9A (0.39) THRBALDH1A1KDM4ECYP1A2CYP2C9
SCHEMBL2292264 0.79 NPC1 (0.44) ALDH1A1KDM4EMAPTLMNARAB9A
SCHEMBL2292578 0.78 KDM4E (0.44) ALDH1A1KDM4EMAPTLMNARAB9A
SCHEMBL2294478 0.78 NPC1 (0.48) MAPTLMNARAB9ANPC1SMN1; SMN2
SCHEMBL5285256 0.78 TP53 (0.48) ALDH1A1KDM4EMAPTHPGDLMNA
SCHEMBL2294510 0.78 SMN1; SMN2 (0.42) ALDH1A1KDM4EMAPTHPGDLMNA
SCHEMBL2294191 0.77 NPC1 (0.38) CYP2C9CYP3A4CYP2C19MAPTLMNA
SCHEMBL5284712 0.77 POLB (0.43) KDM4ESMN1; SMN2
SCHEMBL5280316 0.77 GHSR (0.47) ALDH1A1KDM4ELMNARAB9ANPC1
SCHEMBL2299946 0.77 KMT2A (0.44) ALDH1A1CYP1A2CYP2C9CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828144-A2 INTEGRIN ANTAGONISTS USEFUL AS ANTICANCER AGENTS OSI Pharmaceuticals, Inc. (US) 2007-09-05 EP claimed
WO-2006053342-A2 INTEGRIN ANTAGONISTS USEFUL AS ANTICANCER AGENTS OSI PHARMACEUTICALS, INC. (US) 2006-05-18 WO claimed