SCHEMBL5306277

SCHEMBL5306277

O=C(Nc1cccnn1)c1ccc(N2C=CCN(C(=O)c3cc(F)cc(F)c3C(F)(F)F)C2)nc1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FAAH O00519 9/20 0.37
CRACR2A Q9BSW2 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.33
SCD O00767 2/20 0.32
GLA P06280 1/20 0.32
HTT P42858 1/20 0.32
HDAC2 Q92769 1/20 0.32
EPHX2 P34913 1/20 0.32
SIRT2 Q8IXJ6 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5310018 0.86 SCD (0.45) SCD
SCHEMBL5312568 0.85 FAAH (0.37) FAAHCRACR2AKDM4EALDH1A1SMN1; SMN2
SCHEMBL5306274 0.84 FAAH (0.42) FAAHKDM4ESCDHDAC2
SCHEMBL5312567 0.80 FAAH (0.37) FAAHCRACR2AKDM4EALDH1A1SCD
SCHEMBL5309807 0.78 NPC1 (0.39) CRACR2ASMN1; SMN2SCDGLAHTT
SCHEMBL5311767 0.77 SMN1; SMN2 (0.45) CRACR2AALDH1A1SMN1; SMN2HTTKMT2A
SCHEMBL5309113 0.77 SCD (0.47) SCDKMT2A
SCHEMBL5312273 0.75 KCNQ3 (0.44) KDM4EALDH1A1SMN1; SMN2SCDHTT
SCHEMBL5309408 0.74 SCD (0.47) CRACR2ASCDCYP1A2CYP3A4CYP2D6
SCHEMBL5307080 0.73 SCD (0.40) KDM4EALDH1A1SCDHDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007046867-A2 PIPERIDINE DERIVATIVES AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2007-04-26 WO disclosed