SCHEMBL5307948

SCHEMBL5307948

COc1cccc(Cn2nc(C)c(-c3ccccc3O)c(CCc3cccc(F)c3)c2=O)c1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CASR P41180 9/20 0.49
ALDH1A1 P00352 1/20 0.45
GAA P10253 1/20 0.45
PKM P14618 1/20 0.45
ABCG2 Q9UNQ0 1/20 0.42
PDE5A O76074 1/20 0.42
FPR2 P25090 1/20 0.41
NR1H2 P55055 1/20 0.40
NR1H3 Q13133 1/20 0.40
KDM4E B2RXH2 1/20 0.40
HPGD P15428 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
AURKA O14965 1/20 0.40
AURKB Q96GD4 1/20 0.40
CMA1 P23946 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5315681 0.95 CASR (0.49) CASRALDH1A1GAAPKMABCG2
SCHEMBL5313301 0.93 CASR (0.49) CASRGAAAURKAAURKBPOLB
SCHEMBL5311498 0.92 ALDH1A1 (0.51) CASRALDH1A1GAAPKMABCG2
SCHEMBL5312353 0.90 CASR (0.54) CASRGAAPOLB
SCHEMBL5309465 0.90 CASR (0.47) CASRGAANR1H2NR1H3KDM4E
SCHEMBL5310323 0.89 CASR (0.52) CASRHPGDPOLB
SCHEMBL5308600 0.89 CASR (0.52) CASRABCG2FPR2
SCHEMBL5309931 0.88 CASR (0.47) CASRGAAPOLB
SCHEMBL5310310 0.88 CASR (0.50) CASRALDH1A1KDM4EHPGDPOLB
SCHEMBL5311393 0.88 CASR (0.50) CASRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007044796-A2 PYRIDAZINONE COMPOUNDS AS CALCILYTICS NPS PHARMACEUTICALS, INC. (US) 2007-04-19 WO claimed
WO-2007044796-A2 PYRIDAZINONE COMPOUNDS AS CALCILYTICS NPS PHARMACEUTICALS, INC. (US) 2007-04-19 WO disclosed
WO-2007044796-A2 PYRIDAZINONE COMPOUNDS AS CALCILYTICS NPS PHARMACEUTICALS, INC. (US) 2007-04-19 WO disclosed