SCHEMBL5310264

SCHEMBL5310264

CCCCCN(C)C1(c2ccc(Cl)cc2)CCC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 5/20 0.54
OPRL1 P41146 5/20 0.54
SLC6A4 P31645 5/20 0.45
SLC6A3 Q01959 5/20 0.45
SLC6A2 P23975 3/20 0.45
KCNH2 Q12809 7/20 0.40
CHRM2 P08172 1/20 0.40
ADRA2A P08913 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
HTR2A P28223 1/20 0.40
OPRK1 P41145 1/20 0.40
HTR2B P41595 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
CYP3A4 P08684 1/20 0.40
MAPT P10636 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8605980 0.95 OPRM1 (0.59) OPRM1OPRL1SLC6A4SLC6A3SLC6A2
Hydrochloric Acid SCHEMBL5308781 0.94 OPRM1 (0.57) OPRM1OPRL1SLC6A4SLC6A3SLC6A2
SCHEMBL9765023 0.80 OPRM1 (0.72) OPRM1OPRL1SLC6A4SLC6A3SLC6A2
SCHEMBL8608551 0.79 SLC6A4 (0.50) OPRM1OPRL1SLC6A4SLC6A3SLC6A2
SCHEMBL16887915 0.79 OPRM1 (0.70) OPRM1OPRL1SLC6A4SLC6A3SLC6A2
Hydrochloric Acid SCHEMBL5310523 0.78 CYP3A4 (0.51) OPRM1OPRL1SLC6A4SLC6A3SLC6A2
SCHEMBL16887903 0.77 OPRM1 (0.49) OPRM1OPRL1SLC6A4SLC6A3SLC6A2
Maleic Acid SCHEMBL10899989 0.74 OPRM1 (0.39) OPRM1OPRL1CHRM2LMNACYP3A4
Hydrochloric Acid SCHEMBL5310699 0.74 CYP3A4 (0.54) OPRM1OPRL1SLC6A4SLC6A3SLC6A2
Hydrochloric Acid SCHEMBL2288 0.73 SLC6A3 (0.45) OPRM1OPRL1SLC6A4SLC6A3SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007041677-A9 SOFT TISSUE IMPLANTS AND DRUG COMBINATION COMPOSITIONS, AND USE THEREOF COMBINATORX INC (US) 2007-05-31 WO disclosed
WO-2007041677-A2 SOFT TISSUE IMPLANTS AND DRUG COMBINATION COMPOSITIONS, AND USE THEREOF COMBINATORX, INCORPORATED (US) 2007-04-12 WO disclosed