SCHEMBL5310508

SCHEMBL5310508

COCCn1nc(C)c(-c2ccccc2OCc2ccccc2)c(/C=C/c2cccc(F)c2)c1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
MAOB P27338 2/20 0.36
CYP1A2 P05177 4/20 0.36
CYP3A4 P08684 4/20 0.36
CYP2C9 P11712 3/20 0.36
CASP1 P29466 2/20 0.36
CASP7 P55210 2/20 0.36
HSD17B10 Q99714 2/20 0.36
HPGD P15428 2/20 0.36
CYP2C19 P33261 2/20 0.36
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
ENPP2 Q13822 1/20 0.35
BRD4 O60885 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5310510 1.00 ALDH1A1 (0.40) ALDH1A1MEN1KMT2ASMN1; SMN2LMNA
SCHEMBL5310553 0.93 MEN1 (0.40) ALDH1A1MEN1KMT2ASMN1; SMN2LMNA
SCHEMBL5310556 0.93 MEN1 (0.40) ALDH1A1MEN1KMT2ASMN1; SMN2LMNA
SCHEMBL5308706 0.91 MEN1 (0.37) ALDH1A1MEN1KMT2ASMN1; SMN2LMNA
SCHEMBL5308705 0.91 MEN1 (0.37) ALDH1A1MEN1KMT2ASMN1; SMN2LMNA
SCHEMBL5307926 0.90 ALDH1A1 (0.38) ALDH1A1MEN1KMT2ASMN1; SMN2LMNA
SCHEMBL5307927 0.90 ALDH1A1 (0.38) ALDH1A1MEN1KMT2ASMN1; SMN2LMNA
SCHEMBL5315684 0.90 MEN1 (0.40) ALDH1A1MEN1KMT2ASMN1; SMN2LMNA
SCHEMBL5315689 0.90 MEN1 (0.40) ALDH1A1MEN1KMT2ASMN1; SMN2LMNA
SCHEMBL5311478 0.88 ALDH1A1 (0.40) ALDH1A1MEN1KMT2ASMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007044796-A2 PYRIDAZINONE COMPOUNDS AS CALCILYTICS NPS PHARMACEUTICALS, INC. (US) 2007-04-19 WO disclosed
WO-2007044796-A2 PYRIDAZINONE COMPOUNDS AS CALCILYTICS NPS PHARMACEUTICALS, INC. (US) 2007-04-19 WO disclosed