SCHEMBL5310728

SCHEMBL5310728

C=Cc1c(F)cnc2ccc(OC)cc12.COc1ccc2ncc(F)c(Br)c2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.37
MAPK1 P28482 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
ROCK2 O75116 1/20 0.37
LMNA P02545 2/20 0.36
EGFR P00533 2/20 0.36
GABRA1 P14867 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRA3 P34903 1/20 0.36
GABRA2 P47869 1/20 0.36
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
CYP1A1 P04798 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP1B1 Q16678 1/20 0.35
MAPT P10636 2/20 0.35
GRM1 Q13255 1/20 0.35
HSP90AA1 P07900 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2954867 0.92 KDM4E (0.42) KDM4EMAPK1NPSR1ROCK2LMNA
SCHEMBL2946799 0.88 LMNA (0.43) KDM4EMAPK1NPSR1LMNAEGFR
SCHEMBL5749051 0.81 KDM4E (0.42) KDM4EMAPK1NPSR1ROCK2LMNA
SCHEMBL27632916 0.80 KDM4E (0.41) KDM4EMAPK1NPSR1ROCK2LMNA
SCHEMBL591501 0.79 ALDH1A1 (0.45) KDM4EMAPK1NPSR1LMNAGABRA1
SCHEMBL3831839 0.79 PDE2A (0.30)
SCHEMBL3243876 0.76 SRC (0.43) KDM4EMAPK1NPSR1ROCK2LMNA
SCHEMBL5747019 0.73 PARP1 (0.40) LMNAALDH1A1MAPTHTTTP53
SCHEMBL3273397 0.73 MAP2K1 (0.52) KDM4ENPSR1EGFRMAPTL3MBTL1
SCHEMBL4849696 0.73 KCNH2 (0.41) KDM4EMAPK1NPSR1LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007016610-A2 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2007-02-08 WO disclosed