SCHEMBL5311458

SCHEMBL5311458

COC(=O)C1CCCN1Cc1ccc(Nc2nc3ccc(N(C)c4ccc(F)cc4F)nc3s2)nc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.43
TDO2 P48775 2/20 0.43
GRM2 Q14416 1/20 0.41
ALDH1A1 P00352 3/20 0.35
LCK P06239 1/20 0.35
ITK Q08881 1/20 0.35
GAA P10253 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
DYRK2 Q92630 4/20 0.34
KDM4E B2RXH2 1/20 0.33
TSHR P16473 1/20 0.33
CDK4 P11802 1/20 0.33
CCND1 P24385 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
BMPR1B O00238 1/20 0.32
BMPR1A P36894 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14531000 1.00 IDO1 (0.43) IDO1TDO2GRM2ALDH1A1LCK
SCHEMBL5311790 0.93 IDO1 (0.40) IDO1TDO2GRM2LCKITK
SCHEMBL5311456 0.85 IDO1 (0.44) IDO1TDO2GRM2ALDH1A1LCK
SCHEMBL5316079 0.83 CDK4 (0.40) IDO1TDO2DYRK2CDK4CCND1
SCHEMBL5310039 0.83 FAAH (0.39) DYRK2CDK4
SCHEMBL5315529 0.83 DYRK2 (0.40) DYRK2CDK4CCND1
SCHEMBL5312932 0.82 KDR (0.42) DYRK2CDK4CCND1LTA4H
SCHEMBL5312799 0.81 KDR (0.41) DYRK2CDK4CCND1
SCHEMBL14531377 0.81 DYRK2 (0.40) DYRK2CDK4CCND1
SCHEMBL14531378 0.80 MELK (0.39) GRM2DYRK2CDK4CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007058482-A1 NOVEL INHIBITORS OF PROTEIN KINASE LG LIFE SCIENCES, LTD. (KR) 2007-05-24 WO claimed
WO-2007058482-A1 NOVEL INHIBITORS OF PROTEIN KINASE LG LIFE SCIENCES, LTD. (KR) 2007-05-24 WO disclosed