SCHEMBL531306

SCHEMBL531306

O=C(Nc1ccc(C(O)[C@H](CCn2nnc3ccccc3c2=O)C(=O)O)cc1)c1ccc(C(F)(F)F)cc1F

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GPR139 Q6DWJ6 8/20 0.48
ALDH1A1 P00352 1/20 0.43
AURKA O14965 1/20 0.43
GPR27 Q9NS67 1/20 0.43
KMT2A Q03164 3/20 0.42
KDM4E B2RXH2 1/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.41
HTT P42858 1/20 0.39
MEN1 O00255 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL531305 1.00 GPR139 (0.48) GPR139ALDH1A1AURKAGPR27KMT2A
SCHEMBL529269 0.91 ALDH1A1 (0.46) GPR139ALDH1A1AURKAGPR27KMT2A
SCHEMBL529268 0.91 ALDH1A1 (0.46) GPR139ALDH1A1AURKAGPR27KMT2A
SCHEMBL528620 0.89 ALDH1A1 (0.48) GPR139ALDH1A1KMT2AKDM4EHTT
SCHEMBL528621 0.89 ALDH1A1 (0.48) GPR139ALDH1A1KMT2AKDM4EHTT
SCHEMBL531077 0.85 GPR139 (0.40) GPR139ALDH1A1AURKAGPR27KMT2A
SCHEMBL531078 0.85 GPR139 (0.40) GPR139ALDH1A1AURKAGPR27KMT2A
SCHEMBL526554 0.84 ALDH1A1 (0.52) GPR139ALDH1A1KMT2AKDM4EHTT
SCHEMBL527662 0.84 KMT2A (0.45) GPR139ALDH1A1KMT2AKDM4EHTT
SCHEMBL527661 0.84 KMT2A (0.45) GPR139ALDH1A1KMT2AKDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2598493-A1 MATRIX METALLOPROTEINASE INHIBITORS Ranbaxy Laboratories Limited (IN) 2013-06-05 EP disclosed
WO-2012014114-A1 MATRIX METALLOPROTEINASE INHIBITORS RANBAXY LABORATORIES LIMITED (IN) 2012-02-02 WO disclosed