SCHEMBL531077

SCHEMBL531077

O=C(Nc1ccc(C(O)C(CCn2nnc3ccccc3c2=O)C(=O)N2C(=O)SC[C@@H]2Cc2ccccc2)cc1)c1ccc(C(F)(F)F)cc1F

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GPR139 Q6DWJ6 6/20 0.40
AURKA O14965 3/20 0.36
HTT P42858 2/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35
GPR27 Q9NS67 1/20 0.35
KMT2A Q03164 2/20 0.34
TRPV4 Q9HBA0 1/20 0.34
ALDH1A1 P00352 1/20 0.34
ACKR3 P25106 1/20 0.34
MEN1 O00255 1/20 0.33
RPS6KB1 P23443 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL531078 1.00 GPR139 (0.40) GPR139AURKAHTTKDM4ECYP1A2
SCHEMBL531306 0.85 GPR139 (0.48) GPR139AURKAHTTKDM4EPTGDR2
SCHEMBL531305 0.85 GPR139 (0.48) GPR139AURKAHTTKDM4EPTGDR2
SCHEMBL528378 0.84 KMT2A (0.40) HTTKDM4ESMN1; SMN2KMT2AALDH1A1
SCHEMBL528451 0.81 ALDH1A1 (0.39) GPR139HTTKDM4ESMN1; SMN2KMT2A
SCHEMBL528115 0.81 ALDH1A1 (0.39) GPR139HTTKDM4ESMN1; SMN2KMT2A
SCHEMBL528906 0.79 ALDH1A1 (0.37) GPR139KDM4ESMN1; SMN2KMT2AALDH1A1
SCHEMBL528905 0.79 ALDH1A1 (0.37) GPR139KDM4ESMN1; SMN2KMT2AALDH1A1
SCHEMBL528033 0.77 MMP2 (0.44) GPR139HTTCYP1A2CYP3A4CYP2D6
SCHEMBL528034 0.77 MMP2 (0.44) GPR139HTTCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2598493-A1 MATRIX METALLOPROTEINASE INHIBITORS Ranbaxy Laboratories Limited (IN) 2013-06-05 EP disclosed
WO-2012014114-A1 MATRIX METALLOPROTEINASE INHIBITORS RANBAXY LABORATORIES LIMITED (IN) 2012-02-02 WO disclosed