SCHEMBL5313596

SCHEMBL5313596

Fc1nc(C#Cc2ccc3c(n2)CCCC3)oc1-c1cccnc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
NPY5R Q15761 4/20 0.38
TSHR P16473 3/20 0.33
KDM4E B2RXH2 2/20 0.33
HSD17B10 Q99714 2/20 0.33
HTT P42858 1/20 0.33
GRM5 P41594 6/20 0.33
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
ALDH1A1 P00352 4/20 0.32
LMNA P02545 2/20 0.32
HPGD P15428 2/20 0.32
POLB P06746 1/20 0.32
PKM P14618 1/20 0.32
ALOX15 P16050 1/20 0.32
ALOX12 P18054 1/20 0.32
ATM Q13315 1/20 0.32
MAPK1 P28482 2/20 0.31
CYP1A2 P05177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4322600 0.85 GRM5 (0.48) CYP11B1CYP11B2NPY5RGRM5CYP1A2
SCHEMBL4636436 0.81 ALDH1A1 (0.41) CYP11B1CYP11B2TSHRKDM4EHSD17B10
SCHEMBL4635243 0.77 GRM5 (0.41) HTTGRM5ALDH1A1HPGDCYP2C19
SCHEMBL4330704 0.77 GRM5 (0.53) CYP11B1CYP11B2GRM5
SCHEMBL4322585 0.75 CYP2C19 (0.39) KDM4EHTTGRM5ALDH1A1HPGD
SCHEMBL4335376 0.72 GRM5 (0.59) TSHRKDM4EGRM5ALDH1A1
SCHEMBL28024470 0.68 CYP11B1 (0.55) CYP11B1CYP11B2NPY5RTSHRKDM4E
SCHEMBL4335429 0.65 GRM5 (0.50) CYP11B1CYP11B2KDM4EHSD17B10GRM5
SCHEMBL4328401 0.64 GRM5 (0.63) GRM5
SCHEMBL4330065 0.64 GRM5 (0.48) CYP11B1CYP11B2NPY5RGRM5CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007023242-A1 TETRAHYDROQUINOLINONES AND THEIR USE AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS MERZ PHARMA GMBH & CO. KGAA (DE) 2007-03-01 WO claimed