SCHEMBL5313840

SCHEMBL5313840

O=C1C=c2cc3c(ccc4ccccc43)cc2=CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
HSD17B10 Q99714 3/20 0.47
CYP1B1 Q16678 2/20 0.47
HIF1A Q16665 1/20 0.47
PAX8 Q06710 1/20 0.39
CYP2A6 P11509 1/20 0.39
TSHR P16473 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
CYP1A2 P05177 4/20 0.38
HPGD P15428 2/20 0.38
HPRT1 P00492 3/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
CYP19A1 P11511 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CYP1A1 P04798 1/20 0.33
ERBB2 P04626 1/20 0.33
FYN P06241 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23840 1.00 ALDH1A1 (0.47) ALDH1A1HSD17B10CYP1B1HIF1APAX8
SCHEMBL11515314 0.93 ALDH1A1 (0.41) ALDH1A1HSD17B10CYP1B1HIF1APAX8
SCHEMBL9844906 0.93 CYP1A2 (0.41) ALDH1A1HSD17B10CYP1B1HIF1APAX8
Ethylene Glycol SCHEMBL18525382 0.93 ALDH1A1 (0.41) ALDH1A1HSD17B10CYP1B1HIF1APAX8
SCHEMBL3176812 0.88 ALDH1A1 (0.37) ALDH1A1HSD17B10CYP1B1HIF1APAX8
SCHEMBL31657085 0.87 ALDH1A1 (0.38) ALDH1A1HSD17B10CYP1B1HIF1ATDP1
SCHEMBL31657027 0.87 ALDH1A1 (0.38) ALDH1A1HSD17B10CYP1B1HIF1ATDP1
SCHEMBL31656985 0.87 ALDH1A1 (0.38) ALDH1A1HSD17B10CYP1B1HIF1ATDP1
Trolamine SCHEMBL11041061 0.87 ALDH1A1 (0.36) ALDH1A1HSD17B10CYP1B1HIF1APAX8
Benzanthrone SCHEMBL9018921 0.85 CASP1 (0.49) ALDH1A1HSD17B10CYP1B1HIF1ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1853578-A1 SUBSTITUTED TETRALINS AS SELECTIVE ESTROGEN RECEPTOR-BETA AGONISTS ELI LILLY AND COMPANY (US) 2007-11-14 EP disclosed
WO-2006088716-A1 SUBSTITUTED TETRALINS AS SELECTIVE ESTROGEN RECEPTOR-BETA AGONISTS ELI LILLY AND COMPANY (US) 2006-08-24 WO disclosed