SCHEMBL5314711

SCHEMBL5314711

O=C(NCC1CC1)c1ccc(-c2ccc(C(=O)c3ccccc3C(F)(F)F)nc2)nc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.47
GABRA5 P31644 4/20 0.45
MTTP P55157 1/20 0.45
MAPK14 Q16539 3/20 0.45
CYP2C9 P11712 2/20 0.45
MAPK11 Q15759 1/20 0.44
HDAC4 P56524 2/20 0.44
HPGDS O60760 2/20 0.41
SCD O00767 3/20 0.40
LTC4S Q16873 1/20 0.40
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC7 Q8WUI4 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC10 Q969S8 1/20 0.40
HDAC11 Q96DB2 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC9 Q9UKV0 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5312220 0.88 SCD (0.47) HDAC6MAPK14SCD
SCHEMBL5313199 0.86 HPGDS (0.52) HDAC6GABRA5MAPK14CYP2C9MAPK11
SCHEMBL5312928 0.77 SCD (0.50) HDAC6GABRA5MAPK14SCD
SCHEMBL5312258 0.77 SCD (0.47) SCD
SCHEMBL5307724 0.75 USP30 (0.47) HDAC6SCDHDAC1HDAC8
SCHEMBL1542860 0.73 GABRA5 (0.59) GABRA5MAPK14CYP2C9MAPK11HPGDS
SCHEMBL2295558 0.72 SCD (0.59) GABRA5MAPK14CYP2C9SCD
SCHEMBL5315075 0.71 SCD (0.50) HDAC6GABRA5MAPK14CYP2C9SCD
SCHEMBL5310783 0.71 SCD (0.46) SCD
SCHEMBL5313203 0.71 CNR2 (0.53) SCDLTC4S

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007044085-A2 HETEROARYL COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2007-04-19 WO disclosed