SCHEMBL5315558

SCHEMBL5315558

CC(C)COC(=O)N1CCC(CNC(=O)c2cc(Br)c(N)c3c2OCCC3)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 8/20 0.41
ACHE P22303 2/20 0.40
F2 P00734 1/20 0.36
PLG P00747 1/20 0.36
PRSS1 P07477 1/20 0.36
PRSS2 P07478 1/20 0.36
PRSS3 P35030 1/20 0.36
TPSAB1 Q15661 1/20 0.36
TPSD1 Q9BZJ3 1/20 0.36
TPSG1 Q9NRR2 1/20 0.36
HTR3A P46098 2/20 0.35
HTR3E A5X5Y0 1/20 0.35
HTR3B O95264 1/20 0.35
HTR3D Q70Z44 1/20 0.35
HTR3C Q8WXA8 1/20 0.35
HTR1A P08908 1/20 0.35
ADRA2C P18825 1/20 0.35
PTGS1 P23219 1/20 0.35
ADRA1A P35348 1/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5318285 0.90 HTR4 (0.49) HTR4ACHEHTR3AHTR3EHTR3B
SCHEMBL5318149 0.89 HTR4 (0.41) HTR4ACHEF2PLGPRSS1
SCHEMBL5315555 0.87 KDM4E (0.49) HTR4ACHE
SCHEMBL14382457 0.84 HTR4 (0.44) HTR4ACHEHTR3AHTR3EHTR3B
SCHEMBL17978225 0.80 HTR4 (0.44) HTR4ACHEHTR3AHTR3EHTR3B
SCHEMBL2332701 0.79 HTR4 (0.51) HTR4ACHE
SCHEMBL5316448 0.79 PIM1 (0.45) HTR4HTR3A
Hydrochloric Acid SCHEMBL5631883 0.78 HTR4 (0.50) HTR4ACHE
Hydrochloric Acid SCHEMBL5332277 0.77 HTR4 (0.47) HTR4ACHEHTR3AHTR3EHTR3B
SCHEMBL5318283 0.77 KDM4E (0.49) HTR4ACHEHTR3AHTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007096352-A1 5-AMINO-6-BROMO-N-{ [1- (TETRAHYDR0-2H-PYRAN-4-YLMETHYL) -4-PIPERIDINYL] METHYL}-3, 4 -DIHYDRO-2H-CHROMENE-8-CARBOXAMIDE AS 5-HT4 RECEPTOR AGONIST GLAXO GROUP LIMITED (GB) 2007-08-30 WO disclosed
WO-2007068739-A1 4-AMINO-BENZAMIDE DERIVATIVES AS 5-HT4 RECEPTOR AGONISTS FOR THE TREATMENT OF GASTROINTESTINAL, NEUROLOGICAL AND CARDIOVASCULAR DISORDERS GLAXO GROUP LIMITED (GB) 2007-06-21 WO disclosed