SCHEMBL5316635

SCHEMBL5316635

CC1(C)OB(c2cccc(CN3CCNCC3)c2)OC1(C)C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LPL P06858 1/20 0.51
LIPG Q9Y5X9 1/20 0.51
SIGMAR1 Q99720 1/20 0.49
CXCR4 P61073 5/20 0.41
BRD4 O60885 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP2C9 P11712 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
HIF1A Q16665 1/20 0.40
CHRM3 P20309 5/20 0.39
TDP1 Q9NUW8 2/20 0.39
CHRM2 P08172 1/20 0.39
CHRM1 P11229 1/20 0.39
ADRA2C P18825 1/20 0.39
CCR2 P41597 1/20 0.39
CXCL12 P48061 1/20 0.39
BLM P54132 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1356694 0.88 LPL (0.55) LPLLIPGALDH1A1CYP2C9CYP2C19
SCHEMBL29640063 0.88 LPL (0.55) LPLLIPGALDH1A1CYP2C9CYP2C19
SCHEMBL1641031 0.86 SMN1; SMN2 (0.54) LPLLIPGALDH1A1CYP2C9CYP2C19
SCHEMBL3028131 0.86 LIPG (0.45) LPLLIPGSIGMAR1MEN1KMT2A
Hydrochloric Acid SCHEMBL2072274 0.85 SMN1; SMN2 (0.52) LPLLIPGALDH1A1CYP2C9CYP2C19
SCHEMBL722120 0.85 LPL (0.52) LPLLIPGSIGMAR1BRD4TDP1
SCHEMBL585841 0.85 NCF1 (0.54) LPLLIPGCXCR4BRD4ALDH1A1
Hydrochloric Acid SCHEMBL15845597 0.84 NCF1 (0.52) LPLLIPGCXCR4BRD4ALDH1A1
SCHEMBL15981298 0.83 CXCR4 (0.50) LPLLIPGSIGMAR1CXCR4MEN1
SCHEMBL31341362 0.82 LPL (0.49) LPLLIPGSIGMAR1BRD4CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1812439-A2 KINASE INHIBITORS Takeda San Diego, Inc. (US) 2007-08-01 EP disclosed
WO-2006044687-A2 KINASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-04-27 WO disclosed