SCHEMBL5316749

SCHEMBL5316749

O=C(O)c1nn(C2CCOCC2)c2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 1/20 0.49
HTR4 Q13639 4/20 0.46
CREBBP Q92793 7/20 0.44
CYP3A4 P08684 3/20 0.43
KDM4C Q9H3R0 1/20 0.43
HSD11B1 P28845 1/20 0.42
PIK3CD O00329 2/20 0.41
PIK3R2 O00459 2/20 0.41
PIK3CA P42336 2/20 0.41
PIK3CB P42338 2/20 0.41
PIK3CG P48736 2/20 0.41
PIK3R5 Q8WYR1 2/20 0.41
PIK3R3 Q92569 2/20 0.41
SPR P35270 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
TSHR P16473 1/20 0.38
PMP22 Q01453 1/20 0.38
HIF1A Q16665 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31429395 0.90 CYP3A4 (0.44) SSTR4CYP3A4CYP1A2CYP2D6CYP2C9
SCHEMBL2078485 0.87 HTR3A (0.46) CYP3A4CYP1A2CYP2D6CYP2C9TSHR
SCHEMBL3411552 0.87 KDM4E (0.47)
SCHEMBL8718634 0.86 KDM4E (0.49)
SCHEMBL31195556 0.80 SSTR4 (0.45) SSTR4HTR4CREBBPKDM4CHSD11B1
SCHEMBL25233771 0.78 MEN1 (0.40) CYP3A4CYP1A2CYP2D6CYP2C9TSHR
SCHEMBL15882181 0.77 HTR4 (0.48) HTR4CYP3A4PIK3CDPIK3R2PIK3CA
SCHEMBL31429308 0.77 HTR4 (0.48) HTR4CYP3A4PIK3CDPIK3R2PIK3CA
SCHEMBL31429241 0.76 HTR4 (0.52) HTR4CYP3A4
SCHEMBL15882124 0.76 ROCK1 (0.53) HTR4CYP3A4CYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828179-A2 NICOTINIC ALPHA-7 RECEPTOR LIGANDS AND PREPARATION AND USES THEREOF Memory Pharmaceutical Corporation (US) 2007-09-05 EP disclosed
EP-1745046-A2 1 H-INDAZOLES, BENZOTHIAZOLES, 1,2-BENZIOSOXAZOLES, 1,2-BENZOISOTHIAZOLES, AND CHROMONES AND PREPARATION AND USES THEREOF Memory Pharmaceuticals Corporation (US) 2007-01-24 EP disclosed
WO-2006069097-A2 NICOTINIC ALPHA-7 RECEPTOR LIGANDS AND PREPARATION AND USES THEREOF MEMORY PHARMACEUTICALS CORPORATION (US) 2006-06-29 WO disclosed
WO-2005111038-A2 1H-INDAZOLES, BENZOTHIAZOLES, 1,2-BENZOISOXAZOLES, 1,2-BENZOISOTHIAZOLES, AND CHROMONES AND PREPARATION AND USES THEREOF MEMORY PHARMACEUTICALS CORPORATION (US) 2005-11-24 WO disclosed