SCHEMBL5317013

SCHEMBL5317013

NC(=O)c1ccc(C(=O)CCl)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.64
ALDH1A1 P00352 6/20 0.60
HIF1A Q16665 2/20 0.60
TRPA1 O75762 1/20 0.60
MAPK1 P28482 1/20 0.60
TP53 P04637 1/20 0.52
MAPT P10636 4/20 0.48
POLB P06746 3/20 0.48
RAB9A P51151 1/20 0.48
PARP10 Q53GL7 5/20 0.48
PARP4 Q9UKK3 2/20 0.48
KMT2A Q03164 1/20 0.48
PARP15 Q460N3 1/20 0.48
PARP14 Q460N5 1/20 0.48
PARP16 Q8N5Y8 1/20 0.48
PARP11 Q9NR21 1/20 0.48
PARP1 P09874 2/20 0.48
TSHR P16473 2/20 0.48
CYP3A4 P08684 2/20 0.48
CYP2C19 P33261 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11480265 0.87 GSK3B (0.80) GSK3BALDH1A1HIF1ATRPA1MAPK1
SCHEMBL5317014 0.81 GSK3B (0.64) GSK3BALDH1A1HIF1ATRPA1MAPK1
SCHEMBL10886301 0.80 GSK3B (0.70) GSK3BALDH1A1HIF1ATRPA1MAPK1
Terephthalamide SCHEMBL23774 0.79 PARP1 (0.71) ALDH1A1MAPTPOLBPARP10PARP4
SCHEMBL953871 0.78 GSK3B (1.00) GSK3BALDH1A1HIF1ATRPA1MAPK1
SCHEMBL2968369 0.78 GSK3B (0.67) GSK3BALDH1A1HIF1ATRPA1MAPK1
SCHEMBL5787064 0.78 GSK3B (0.67) GSK3BALDH1A1HIF1ATRPA1MAPK1
SCHEMBL22919688 0.78 PARP10 (0.50) ALDH1A1MAPTPOLBPARP10PARP4
SCHEMBL6266724 0.78 ALDH1A1 (0.70) GSK3BALDH1A1HIF1ATRPA1MAPK1
SCHEMBL3376212 0.78 PARP10 (0.50) ALDH1A1MAPTPOLBPARP10PARP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103957711-A use of substituted isoquinolinones, isoquinolinediones, isoquinolinetriones and dihydroisoquinolinones or their respective salts as active agents against abiotic stress in plants BAYER IP GMBH 2014-07-30 CN disclosed
WO-2007067993-A1 INHIBITORS OF HISTONE DEACETYLASE FOR THE TREATMENT OF DISEASE KALYPSYS, INC. (US) 2007-06-14 WO disclosed