SCHEMBL5317286

SCHEMBL5317286

O=C(O)N1CCN(c2cnc3ccccc3c2)CC1

nearest known ligand 0.70

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.70
HTR3A P46098 1/20 0.65
DRD3 P35462 2/20 0.56
DRD2 P14416 1/20 0.56
CHRNB2 P17787 1/20 0.56
CHRNA4 P43681 1/20 0.56
DHFR P00374 1/20 0.55
CCKAR P32238 11/20 0.53
HTR2A P28223 1/20 0.50
HTR2C P28335 1/20 0.50
TSHR P16473 1/20 0.49
MGAM O43451 1/20 0.49
HDAC1 Q13547 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20274184 0.85 AKR1C3 (0.66) AKR1C3HTR3ADRD3DRD2CHRNB2
SCHEMBL14783389 0.83 AKR1C3 (0.51) AKR1C3HTR3ADRD3DRD2CHRNB2
Oxalic Acid SCHEMBL8147179 0.83 CHRNB2 (0.63) AKR1C3HTR3ADRD3DRD2CHRNB2
SCHEMBL31254486 0.81 AKR1C3 (0.61) AKR1C3HTR3ADHFRCCKAR
SCHEMBL4054998 0.81 AKR1C3 (0.61) AKR1C3HTR3ADHFRCCKAR
SCHEMBL5800979 0.81 HTR3A (0.58) AKR1C3HTR3ADRD3DRD2CHRNB2
SCHEMBL14784331 0.80 MAPT (0.48) AKR1C3CCKAR
SCHEMBL28537114 0.79 HTR3A (0.68) AKR1C3HTR3ADRD3DRD2CHRNB2
Trifluoroacetic Acid SCHEMBL4522904 0.79 HTR3A (0.76) AKR1C3HTR3ADRD3DRD2CHRNB2
SCHEMBL14783547 0.79 AKR1C3 (0.47) AKR1C3HTR3ADRD3DRD2CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828154-A1 PHENYL-PIPERAZIN METHANONE DERIVATIVES F. Hoffmann-Roche AG (CH) 2007-09-05 EP disclosed
WO-2006061135-A1 PHENYL-PIPERAZIN METHANONE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2006-06-15 WO disclosed