SCHEMBL5317475

SCHEMBL5317475

COc1ccc(NC(N)=O)c(OC)c1

nearest known ligand 0.71

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.71
CYP1A1 P04798 1/20 0.65
CYP1A2 P05177 1/20 0.65
CYP1B1 Q16678 1/20 0.65
HPGD P15428 1/20 0.65
MAPT P10636 3/20 0.63
NPC1 O15118 3/20 0.62
RAB9A P51151 3/20 0.62
MEN1 O00255 3/20 0.62
KMT2A Q03164 3/20 0.62
SMN1; SMN2 Q16637 2/20 0.62
GAA P10253 2/20 0.61
LMNA P02545 1/20 0.61
AHR P35869 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29757951 1.00 ALDH1A1 (0.71) ALDH1A1CYP1A1CYP1A2CYP1B1HPGD
SCHEMBL167053 0.86 GAA (0.67) ALDH1A1HPGDMAPTNPC1RAB9A
SCHEMBL18415558 0.86 ALDH1A1 (0.75) ALDH1A1CYP1A1CYP1A2CYP1B1HPGD
SCHEMBL5833241 0.84 ALDH1A1 (0.73) ALDH1A1CYP1A1CYP1A2CYP1B1HPGD
SCHEMBL30622065 0.84 HSD17B1 (0.75) ALDH1A1CYP1A1CYP1A2CYP1B1HPGD
SCHEMBL11660515 0.84 ALDH1A1 (0.73) ALDH1A1CYP1A1CYP1A2CYP1B1HPGD
SCHEMBL2191052 0.84 HSD17B1 (0.75) ALDH1A1CYP1A1CYP1A2CYP1B1HPGD
SCHEMBL4634999 0.84 NPC1 (0.59) ALDH1A1CYP1A1CYP1A2CYP1B1HPGD
SCHEMBL30945495 0.83 ALDH1A1 (0.61) ALDH1A1CYP1A1CYP1A2CYP1B1HPGD
SCHEMBL10506942 0.83 EPHX1 (0.61) ALDH1A1HPGDMAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1845978-A1 SUBSTITUTED PYRAZOLO-PYRIDINES, COMPOSITIONS CONTAINING THEM, METHOD FOR THE PRODUCTION THEREOF, AND THEIR USE Aventis Pharma S.A. (FR) 2007-10-24 EP disclosed
WO-2006077319-A1 SUBSTITUTED PYRAZOLO-PYRIDINES, COMPOSITIONS CONTAINING THEM, METHOD FOR THE PRODUCTION THEREOF, AND THEIR USE AVENTIS PHARMA S.A. (FR) 2006-07-27 WO disclosed
US-5780483-A IL-8 receptor antagonists SMITHKLINE BEECHAM CORPORATION (US) 1998-07-14 US disclosed