SCHEMBL5318145

SCHEMBL5318145

[CH2]CN(C)C(=O)c1ccc(C#N)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 2/20 0.60
GSK3B P49841 2/20 0.47
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.47
NPC1 O15118 1/20 0.47
ALDH1A1 P00352 2/20 0.45
MAPT P10636 2/20 0.45
MLYCD O95822 1/20 0.43
TSHR P16473 1/20 0.41
TMEM97 Q5BJF2 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
TP53 P04637 2/20 0.41
PDK1 Q15118 1/20 0.41
PDK2 Q15119 1/20 0.41
PDK3 Q15120 1/20 0.41
PDK4 Q16654 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL123989 0.83 NSD2 (0.42) NSD2ALDH1A1MLYCDHPGD
SCHEMBL5317404 0.81 NSD2 (0.58) NSD2GSK3BCA1CA2KMT2A
SCHEMBL10933810 0.80 NSD2 (0.55) NSD2GSK3BCA1CA2KMT2A
SCHEMBL13151106 0.78 NSD2 (0.54) NSD2GSK3BCA1CA2KMT2A
SCHEMBL7533635 0.77 ALDH1A1 (0.55) KMT2AMEN1NPC1ALDH1A1MAPT
SCHEMBL6796753 0.76 NSD2 (0.77) NSD2CA2KMT2AMEN1NPC1
SCHEMBL294286 0.76 KMT2A (0.53) KMT2AMEN1ALDH1A1MAPTMLYCD
SCHEMBL23015300 0.75 NSD2 (1.00) NSD2KMT2AMEN1NPC1ALDH1A1
SCHEMBL5414969 0.75 NSD2 (0.52) NSD2GSK3BCA1CA2KMT2A
SCHEMBL7236313 0.75 NSD2 (0.71) NSD2KMT2AMEN1NPC1MLYCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007069986-A1 NEW OXABISPIDINE COMPOUNDS FOR THE TREATMENT OF CARDIAC ARRHYTHMIAS ASTRAZENECA AB (SE) 2007-06-21 WO claimed
WO-2007069986-A1 NEW OXABISPIDINE COMPOUNDS FOR THE TREATMENT OF CARDIAC ARRHYTHMIAS ASTRAZENECA AB (SE) 2007-06-21 WO disclosed