SCHEMBL5318243

SCHEMBL5318243

Cc1cc(Cl)ccc1Cn1nc(-c2nnn[nH]2)c2ccc(C(F)(F)F)cc21

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 1/20 0.36
PDE5A O76074 3/20 0.35
PTGER1 P34995 1/20 0.35
NR1H2 P55055 4/20 0.34
NR1H3 Q13133 4/20 0.34
SLC22A12 Q96S37 1/20 0.34
HTT P42858 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
PTGDR2 Q9Y5Y4 2/20 0.32
BUB1 O43683 1/20 0.32
AKR1B1 P15121 1/20 0.32
GCGR P47871 1/20 0.32
POLB P06746 1/20 0.31
GUCY1A1 Q02108 1/20 0.31
GUCY1B1 Q02153 1/20 0.31
KCNA3 P22001 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5320369 0.90 NR1H2 (0.43) PDE5APTGER1NR1H2NR1H3GUCY1A1
SCHEMBL2889462 0.84 CYP1A2 (0.43) PDE5ABUB1POLB
SCHEMBL5321077 0.84 NR1H2 (0.42) PDE5APTGER1NR1H2NR1H3SLC22A12
SCHEMBL5317498 0.83 CCR2 (0.36) CCR2NR1H2NR1H3SLC22A12HTT
SCHEMBL5318688 0.79 AKR1B1 (0.36) CCR2NR1H2NR1H3SLC22A12PTGDR2
SCHEMBL4097771 0.75 CYP1A2 (0.54) CCR2PTGER1SLC22A12PTGDR2AKR1B1
SCHEMBL5270492 0.75 AKR1B1 (0.39) CCR2PTGER1NR1H2NR1H3SLC22A12
SCHEMBL5322124 0.74 AKR1B1 (0.54) SLC22A12PTGDR2AKR1B1
SCHEMBL5322328 0.74 ENPP2 (0.41) CCR2PTGER1NR1H2NR1H3SLC22A12
SCHEMBL5318544 0.74 AKR1B1 (0.38) CCR2PTGER1NR1H2NR1H3SLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1786424-A2 LONIDAMINE ANALOGUES AND THEIR USE IN MALE CONTRACEPTION AND CANCER TREATMENT The University of Kansas (US) 2007-05-23 EP claimed
WO-2006023704-A2 LONIDAMINE ANALOGUES AND THEIR USE IN MALE CONTRACEPTION AND CANCER TREATMENT UNIVERSITY OF KANSAS (US) 2006-03-02 WO claimed