SCHEMBL5318329

SCHEMBL5318329

CCN1CCC(N(CC)C(=O)c2ccc3c(c2)nc(NC2CCCC2)n3C)CC1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ITK Q08881 11/20 0.51
KCNH2 Q12809 1/20 0.44
RAF1 P04049 1/20 0.43
BRAF P15056 1/20 0.43
HRH3 Q9Y5N1 1/20 0.40
CNR2 P34972 2/20 0.40
BCHE P06276 1/20 0.40
BRD4 O60885 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
KDM4E B2RXH2 1/20 0.39
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5317039 0.85 ITK (0.46) ITKHRH3CNR2BCHEBRD4
SCHEMBL5315592 0.81 ITK (0.53) ITK
SCHEMBL5315730 0.78 ITK (0.46) ITKHRH3CNR2BCHEBRD4
SCHEMBL5318291 0.76 L3MBTL1 (0.54) KCNH2RAF1BRAFHDAC6
SCHEMBL5317065 0.76 JAK2 (0.47) ITKHRH3CNR2
SCHEMBL5317545 0.74 ITK (0.44) ITKCNR2
SCHEMBL5318216 0.73 ITK (0.43) ITKCNR2BCHEKDM4E
SCHEMBL5315360 0.73 ITK (0.43) ITKCNR2
SCHEMBL5315400 0.72 FLT3 (0.48) ITK
SCHEMBL5318313 0.69 ITK (0.47) ITKHRH3CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007069053-A1 BENZIMIDAZOLE ANTAGONISTS OF THE H-3 RECEPTOR PFIZER PRODUCTS INC. (US) 2007-06-21 WO claimed
WO-2007069053-A1 BENZIMIDAZOLE ANTAGONISTS OF THE H-3 RECEPTOR PFIZER PRODUCTS INC. (US) 2007-06-21 WO disclosed