SCHEMBL5318595

SCHEMBL5318595

O=C(O)N1CC(NOCc2ccccc2)c2ccccc2N1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
IDO1 P14902 4/20 0.36
TDO2 P48775 2/20 0.36
HTR1A P08908 2/20 0.35
SLC6A2 P23975 2/20 0.35
SLC6A4 P31645 2/20 0.35
SLC6A3 Q01959 2/20 0.35
S1PR5 Q9H228 1/20 0.35
EPHX2 P34913 1/20 0.34
TNKS2 Q9H2K2 1/20 0.34
MMP13 P45452 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
HTR2C P28335 1/20 0.34
EGFR P00533 1/20 0.34
SRC P12931 1/20 0.34
GAA P10253 1/20 0.34
MAPK1 P28482 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4862019 0.86 MEN1 (0.37) IDO1ALDH1A1MAPTMAPK1
SCHEMBL5322672 0.79 CASP1 (0.37) MAPTGAAMAPK1SMN1; SMN2
SCHEMBL5254943 0.75 NPC1 (0.38) NPC1RAB9AS1PR5EPHX2ALDH1A1
SCHEMBL5187275 0.72 GPR183 (0.39) NPC1RAB9AALDH1A1MAPT
SCHEMBL5270565 0.71 SLC6A2 (0.37) NPC1RAB9AIDO1TDO2HTR1A
Hydrochloric Acid SCHEMBL4865376 0.70 SLC6A2 (0.36) NPC1RAB9AIDO1TDO2HTR1A
SCHEMBL5330841 0.68 TSHR (0.40) NPC1RAB9AHTR1ASLC6A2SLC6A4
SCHEMBL4697074 0.68 NPC1 (0.34) NPC1RAB9AS1PR5EPHX2ALDH1A1
SCHEMBL5187221 0.66 NPC1 (0.37) NPC1RAB9AEPHX2ALDH1A1MAPT
SCHEMBL3305431 0.65 LMNA (0.34) NPC1RAB9AS1PR5EPHX2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537117-B1 BENZOTRIAZABICYCLIC DERIVATIVES AND USE THEREOF AS BETA-LACTAMASE INHIBITORS AND ANTI-BACTERIAL AGENTS AVENTIS PHARMA SA (FR) 2007-01-17 EP disclosed