SCHEMBL7464584

SCHEMBL7464584

Clc1ccc2c(c1)c1c(n2Cc2ccccc2)CCCC1

nearest known ligand 0.67

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.67
CA2 P00918 3/20 0.67
PTGS1 P23219 1/20 0.62
PTGS2 P35354 1/20 0.62
HTR6 P50406 2/20 0.59
FABP4 P15090 3/20 0.58
SLC2A1 P11166 2/20 0.52
NPC1 O15118 1/20 0.52
LMNA P02545 1/20 0.52
HTT P42858 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
FABP3 P05413 1/20 0.51
HDAC1 Q13547 1/20 0.51
HDAC10 Q969S8 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3857256 0.85 CA1 (0.65) CA1CA2PTGS1PTGS2HTR6
SCHEMBL6045346 0.84 CA1 (0.94) CA1CA2HTR6FABP4HDAC1
SCHEMBL31554283 0.82 FABP4 (0.59) PTGS1PTGS2FABP4FABP3
SCHEMBL3853296 0.81 CA1 (0.59) CA1CA2PTGS1PTGS2HTR6
SCHEMBL6925477 0.79 PTGS1 (0.65) CA1CA2PTGS1PTGS2FABP4
SCHEMBL3859121 0.78 HTR6 (0.67) CA1CA2PTGS1PTGS2HTR6
SCHEMBL3318218 0.78 PTGS1 (0.53) CA1CA2PTGS1PTGS2HTR6
SCHEMBL27568575 0.77 PTGDR2 (0.69)
Acetic Acid SCHEMBL9518648 0.77 CA1 (0.78) CA1CA2HTR6FABP4FABP3
SCHEMBL5319783 0.76 PTGS1 (0.48) CA1CA2PTGS1PTGS2HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1058678-B1 METAL-CATALYZED ARYLATIONS AND VINYLATIONS OF HYDRAZINES, HYDRAZONES, HYDROXYLAMINES AND OXIMES MASSACHUSETTS INST TECHNOLOGY (US) 2002-12-11 EP disclosed
US-6465693-B2 TRANSITION METAL CATALYZED ARYLATION OR VINYLATION; COMBINATORIAL CHEMISTRY MASSACHUSETTS INSTITUTE OF TECHNOLOGY 2002-10-15 US disclosed
US-20010031894-A1 Metal-catalyzed arylations of hydrazines, hydrazones, and related substrates BUCHWALD STEPHEN L (US) 2001-10-18 US disclosed
US-6235936-B1 TRANSITION METAL CATALYST FOR ARYLATION MASSACHUSETTS INSTITUTE OF TECHNOLOGY 2001-05-22 US disclosed
EP-1058678-A2 METAL-CATALYZED ARYLATIONS AND VINYLATIONS OF HYDRAZINES, HYDRAZONES, HYDROXYLAMINES AND OXIMES Massachusetts Institute of Technology (US) 2000-12-13 EP disclosed
WO-1999043643-A2 METAL-CATALYZED ARYLATIONS AND VINYLATIONS OF HYDRAZINES, HYDRAZONES, HYDROXYLAMINES AND OXIMES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1999-09-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010031894-A1 Metal-catalyzed arylations of hydrazines, hydrazones, and related substrates IDO1, IDO2, AHR CA1 749/4885CA2 288/4885PTGS1 2384/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.