SCHEMBL5320166

SCHEMBL5320166

CC1(C)Cc2cc([AsH]c3ccc(F)cc3F)ccc2C1=O

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32
MALT1 Q9UDY8 1/20 0.32
GRM1 Q13255 1/20 0.31
MAPK14 Q16539 1/20 0.31
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20951663 0.80 CA1 (0.43) TDP2ALDH1A1CA1CA2CA7
SCHEMBL5288032 0.72 MAPK14 (0.56) ALDH1A1MAPK14
SCHEMBL2390689 0.71 ACHE (0.46) TDP2ALDH1A1CA1CA2CA7
SCHEMBL14430335 0.67 HTT (0.33) GRM1
SCHEMBL12310527 0.66 METAP1 (0.44) ALDH1A1CA1CA2CA7CA9
SCHEMBL9589413 0.65 SRD5A1 (0.45) CA1CA2CA7CA9MALT1
SCHEMBL10908106 0.65 CA1 (0.41) TDP2ALDH1A1CA1CA2CA7
SCHEMBL14430356 0.65 ABCC9 (0.32) GRM1
SCHEMBL30701788 0.65 ABCC9 (0.32) GRM1
SCHEMBL5293741 0.65 MAPK14 (0.58) MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007000337-A1 BICYCLIC DERIVATIVES AS P38 KINASE INHIBITORS PALAU PHARMA, S.A. (ES) 2007-01-04 WO disclosed