SCHEMBL532041

SCHEMBL532041

Cc1cc(C)c(N2CCCC2)c(C)c1NS(=O)(=O)NC(=O)Cc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.42
KMT2A Q03164 4/20 0.42
MAPT P10636 3/20 0.42
MEN1 O00255 3/20 0.42
KDM4E B2RXH2 2/20 0.42
USP2 O75604 1/20 0.42
POLB P06746 1/20 0.42
HPGD P15428 1/20 0.42
BLM P54132 1/20 0.42
KCNQ2 O43526 2/20 0.42
GAA P10253 2/20 0.42
NR4A1 P22736 1/20 0.42
PKM P14618 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
BRPF1 P55201 2/20 0.41
CNR2 P34972 2/20 0.40
SLC2A1 P11166 1/20 0.40
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL532946 0.84 KCNQ2 (0.53) ALDH1A1KMT2AMAPTMEN1KDM4E
SCHEMBL532988 0.80 ALDH1A1 (0.42) ALDH1A1KMT2AKDM4EPOLBHPGD
SCHEMBL533164 0.78 PTGES2 (0.39) KMT2AMEN1POLB
SCHEMBL532776 0.77 FFAR4 (0.54) ALDH1A1KMT2AMAPTMEN1POLB
SCHEMBL532980 0.73 JAK2 (0.48) ALDH1A1KMT2AMAPTMEN1KDM4E
SCHEMBL533170 0.73 S100A9 (0.43) KCNQ2
SCHEMBL534077 0.73 TSHR (0.47) ALDH1A1KMT2AMAPTMEN1POLB
SCHEMBL533059 0.72 MEN1 (0.55) ALDH1A1KMT2AMAPTMEN1KDM4E
SCHEMBL533006 0.72 HTR6 (0.43) ALDH1A1KMT2AMAPTMEN1KDM4E
SCHEMBL533083 0.71 EDNRA (0.46) ALDH1A1MAPTPOLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2415760-A2 CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2012-02-08 EP disclosed
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed