SCHEMBL5320832

SCHEMBL5320832

O=C(O)C(C(=O)O)=C(c1ccc(Cl)cc1)c1ccc(Cl)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.58
ALOX15 P16050 1/20 0.58
CES2 O00748 3/20 0.54
CES1 P23141 3/20 0.54
L3MBTL1 Q9Y468 3/20 0.52
MAPK1 P28482 2/20 0.52
CYP3A4 P08684 1/20 0.52
ATM Q13315 1/20 0.52
SRD5A2 P31213 1/20 0.52
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
ERCC5 P28715 1/20 0.50
FEN1 P39748 1/20 0.50
GSK3B P49841 2/20 0.46
MAPT P10636 2/20 0.45
ALDH1A1 P00352 2/20 0.45
KDM4E B2RXH2 1/20 0.45
LMNA P02545 1/20 0.45
NR4A1 P22736 1/20 0.44
CYP19A1 P11511 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4619034 0.87 TSHR (0.56) TSHRALOX15CES2CES1L3MBTL1
SCHEMBL2782261 0.77 CES1 (0.52) TSHRALOX15CES2CES1L3MBTL1
SCHEMBL27938664 0.76 TSHR (0.72) TSHRALOX15CES2CES1L3MBTL1
SCHEMBL927606 0.75 CES2 (0.75) TSHRALOX15CES2CES1L3MBTL1
4-Chloro-Benzoic Acid SCHEMBL9194331 0.75 TSHR (0.90) TSHRALOX15CES2CES1SRD5A2
SCHEMBL15180838 0.75 CES2 (0.75) TSHRALOX15CES2CES1L3MBTL1
SCHEMBL5451212 0.74 HPGD (0.48) TSHRALOX15CES2CES1L3MBTL1
4-Chloro-Benzoic Acid SCHEMBL28384 0.74 TSHR (1.00) TSHRALOX15CES2CES1SRD5A2
4-Chloro-Benzoic Acid SCHEMBL1331727 0.74 TSHR (1.00) TSHRALOX15CES2CES1SRD5A2
SCHEMBL17802344 0.73 CES2 (0.59) TSHRALOX15CES2CES1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007128672-A1 SUBSTITUTED HEXAHYDRO-1,4-DIAZEPIN-5-ONES AND COMPOSITIONS STABILIZED THEREWITH CIBA HOLDING INC. (CH) 2007-11-15 WO disclosed