SCHEMBL5320962

SCHEMBL5320962

O=C1N(Cc2ccccc2)N=C(C2CCCCC2)c2ccccc2N1Cc1cccc([N+](=O)[O-])c1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTH1R Q03431 8/20 0.56
ALDH1A1 P00352 1/20 0.53
HPGD P15428 1/20 0.53
HTT P42858 1/20 0.53
CCKBR P32239 10/20 0.47
CCKAR P32238 4/20 0.46
CASP1 P29466 1/20 0.44
CASP3 P42574 1/20 0.44
CASP4 P49662 1/20 0.44
CASP7 P55210 1/20 0.44
CASP9 P55211 1/20 0.44
CASP6 P55212 1/20 0.44
CASP8 Q14790 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5320618 0.92 PTH1R (0.55) PTH1RALDH1A1CCKBRCCKARCASP1
SCHEMBL5320334 0.83 PTH1R (0.69) PTH1RALDH1A1CCKBR
SCHEMBL5323577 0.80 PTH1R (0.47) PTH1RALDH1A1CCKBRCCKARCASP1
SCHEMBL5320380 0.77 PTH1R (0.57) PTH1RHPGDHTTCCKBR
SCHEMBL5324664 0.76 PTH1R (0.58) PTH1RCCKBRCASP1CASP3CASP4
SCHEMBL5321708 0.76 PTH1R (0.56) PTH1RALDH1A1CASP1CASP3CASP4
SCHEMBL5322971 0.74 PTH1R (0.54) PTH1RCCKBRCASP1CASP3CASP4
SCHEMBL5327910 0.74 PTH1R (0.56) PTH1RCCKBR
SCHEMBL5280948 0.73 PTH1R (0.76) PTH1RCCKBRCCKAR
SCHEMBL5325678 0.73 PTH1R (0.57) PTH1RCASP1CASP3CASP4CASP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129120-A9 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2007-03-22 WO disclosed
WO-2006129120-A2 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2006-12-07 WO disclosed