SCHEMBL5323904

SCHEMBL5323904

Nc1cc(C(=O)N2CCC(Oc3ccc(F)cc3)CC2)c(Cl)cn1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.48
TRPC6 Q9Y210 5/20 0.48
ADRB2 P07550 1/20 0.47
PRKAA2 P54646 3/20 0.46
HRH1 P35367 2/20 0.44
CCR3 P51677 2/20 0.44
MLNR O43193 1/20 0.44
CYP3A4 P08684 1/20 0.44
KCNH2 Q12809 1/20 0.44
MCHR1 Q99705 1/20 0.44
CNR1 P21554 1/20 0.43
HSD11B1 P28845 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5318563 0.84 EPHX2 (0.52) EPHX2ADRB2HRH1CCR3MLNR
SCHEMBL14466887 0.83 PRKAA2 (0.49) EPHX2ADRB2PRKAA2HRH1CCR3
SCHEMBL5317962 0.83 HPGD (0.50) EPHX2ADRB2HRH1CCR3MLNR
SCHEMBL5342932 0.80 ADRB2 (0.47) EPHX2ADRB2PRKAA2HRH1CCR3
SCHEMBL5321693 0.80 EPHX2 (0.49) EPHX2ADRB2HRH1CCR3MLNR
SCHEMBL14467022 0.79 EPHX2 (0.44) EPHX2ADRB2PRKAA2HRH1CCR3
SCHEMBL14466895 0.76 PRKAA2 (0.51) EPHX2ADRB2PRKAA2HRH1CCR3
SCHEMBL5323864 0.74 MAPK14 (0.49) EPHX2ADRB2HRH1CCR3MLNR
SCHEMBL1809345 0.74 ADRB2 (0.71) ADRB2HRH1HSD11B1
SCHEMBL1809547 0.73 EPHX2 (0.52) EPHX2ADRB2HRH1CCR3MLNR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007082079-A2 PIPERIDINE AMIDE DERIVATIVES AS PROTEIN KINASE INHIBITORS THE SCRIPPS RESEARCH INSTITUTE (US) 2007-07-19 WO disclosed