Eperezolid

Eperezolid

SCHEMBL5325217

CC(=O)NC[C@H]1CN(c2ccc(N3CCN(C(=O)CO)CC3)c(F)c2)C(=O)O1.N

nearest known ligand 0.75

Full drug profile on Sugi Atlas →

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAOB P27338 7/20 0.75
MAOA P21397 5/20 0.75
PTGS1 P23219 2/20 0.75
SDHA P31040 2/20 0.75
LMNA P02545 1/20 0.75
CALML3 P27482 1/20 0.75
F10 P00742 6/20 0.72

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Eperezolid SCHEMBL1176950 0.99 MAOB (0.76) MAOBMAOAPTGS1SDHALMNA
Eperezolid SCHEMBL186562 0.99 MAOB (0.76) MAOBMAOAPTGS1SDHALMNA
Eperezolid SCHEMBL29421647 0.99 MAOB (0.76) MAOBMAOAPTGS1SDHALMNA
Eperezolid SCHEMBL5328753 0.96 F10 (0.71) MAOBMAOAPTGS1SDHALMNA
Eperezolid SCHEMBL7497950 0.95 MAOB (0.85) MAOBMAOAPTGS1SDHALMNA
SCHEMBL6160243 0.93 F10 (0.72) MAOBMAOAPTGS1SDHALMNA
SCHEMBL6160239 0.93 F10 (0.72) MAOBMAOAPTGS1SDHALMNA
SCHEMBL4163039 0.93 MAOA (0.67) MAOBMAOAPTGS1SDHALMNA
SCHEMBL10151505 0.92 MAOB (0.76) MAOBMAOAPTGS1SDHALMNA
SCHEMBL12674054 0.91 MAOB (0.73) MAOBMAOAPTGS1SDHALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007138381-A2 PHOSPHONATED OXAZOLIDINONES AND USES THEREOF FOR THE PREVENTION AND TREATMENT OF BONE AND JOINT INFECTIONS TARGANTA THERAPEUTICS INC. (CA) 2007-12-06 WO claimed
WO-2007138381-A2 PHOSPHONATED OXAZOLIDINONES AND USES THEREOF FOR THE PREVENTION AND TREATMENT OF BONE AND JOINT INFECTIONS TARGANTA THERAPEUTICS INC. (CA) 2007-12-06 WO disclosed