SCHEMBL5325791

SCHEMBL5325791

COc1ccc(Oc2c(Cl)cc(N3C(=O)CNC3=O)cc2Cl)cc1Cc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.41
THRB P10828 4/20 0.40
RORC P51449 3/20 0.40
THRA P10827 1/20 0.37
AADAT Q8N5Z0 1/20 0.37
NPBWR1 P48145 4/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
SIGMAR1 Q99720 1/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5325839 0.89 PDE4A (0.37) CYP3A4THRBTHRAAADATMEN1
SCHEMBL5326880 0.88 RORC (0.38) CYP3A4THRBRORCNPBWR1MEN1
SCHEMBL5333107 0.86 THRB (0.50) CYP3A4THRBTHRAMEN1KMT2A
SCHEMBL5326116 0.83 THRB (0.39) CYP3A4THRBRORCTHRANPBWR1
SCHEMBL5325788 0.81 THRB (0.40) CYP3A4THRBRORCTHRAAADAT
SCHEMBL5323878 0.79 RORC (0.55) THRBRORCTHRA
SCHEMBL5329553 0.79 ESRRA (0.39) THRBRORCTHRANPBWR1MEN1
SCHEMBL5326865 0.78 RORC (0.46) THRBRORCTHRANPBWR1MEN1
SCHEMBL16496798 0.77 CYP1A2 (0.46) THRBRORCNPBWR1MEN1KMT2A
SCHEMBL5324548 0.77 POLB (0.56) NPBWR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007132475-A1 SELECTIVE TR-BETA 1 AGONIST CADILA HEALTHCARE LIMITED (IN) 2007-11-22 WO claimed
WO-2007132475-A1 SELECTIVE TR-BETA 1 AGONIST CADILA HEALTHCARE LIMITED (IN) 2007-11-22 WO disclosed