SCHEMBL5325839

SCHEMBL5325839

COc1ccc(Oc2c(Br)cc(N3C(=O)CNC3=O)cc2Br)cc1Cc1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
THRA P10827 2/20 0.37
THRB P10828 2/20 0.37
AADAT Q8N5Z0 1/20 0.37
PDE10A Q9Y233 1/20 0.35
TRIM24 O15164 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
POLB P06746 1/20 0.34
GAA P10253 1/20 0.34
SIGMAR1 Q99720 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5325791 0.89 CYP3A4 (0.41) PDE4APDE4BPDE4CPDE4DTHRA
SCHEMBL5325834 0.81 PDE4A (0.37) PDE4APDE4BPDE4CPDE4DTHRA
SCHEMBL2170953 0.77 TTR (0.44) THRATHRBMEN1KMT2A
SCHEMBL5326880 0.76 RORC (0.38) THRBMEN1KMT2APOLBGAA
SCHEMBL5333107 0.74 THRB (0.50) THRATHRBMEN1KMT2ACYP3A4
SCHEMBL16495779 0.72 ALDH1A1 (0.52) THRATHRBMEN1KMT2APOLB
SCHEMBL16495780 0.72 ALDH1A1 (0.52) THRATHRBMEN1KMT2APOLB
SCHEMBL5325788 0.69 THRB (0.40) PDE4APDE4BPDE4CPDE4DTHRA
SCHEMBL11288852 0.68 LTA4H (0.58)
SCHEMBL18932876 0.68 THRB (0.45) THRBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007132475-A1 SELECTIVE TR-BETA 1 AGONIST CADILA HEALTHCARE LIMITED (IN) 2007-11-22 WO claimed
WO-2007132475-A1 SELECTIVE TR-BETA 1 AGONIST CADILA HEALTHCARE LIMITED (IN) 2007-11-22 WO disclosed