SCHEMBL5325876

SCHEMBL5325876

CCOC(=O)c1ccc2ncc(C(=O)OCC)c(Nc3cccc(C(C)=O)c3)c2c1

nearest known ligand 0.93

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.81
CREBBP Q92793 1/20 0.79
KDM4E B2RXH2 3/20 0.78
ALDH1A1 P00352 3/20 0.78
PKM P14618 1/20 0.78
MAPT P10636 7/20 0.69
SMN1; SMN2 Q16637 2/20 0.68
RXFP1 Q9HBX9 1/20 0.68
PAX8 Q06710 1/20 0.65
AURKB Q96GD4 6/20 0.62
AURKA O14965 4/20 0.62
LMNA P02545 2/20 0.61
POLB P06746 1/20 0.61
GAA P10253 1/20 0.61
MAPK1 P28482 1/20 0.61
MC4R P32245 1/20 0.61
HTT P42858 1/20 0.61
CLK1 P49759 1/20 0.61
GSK3A P49840 1/20 0.61
GSK3B P49841 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5323732 0.96 CREBBP (0.86) TP53CREBBPKDM4EALDH1A1PKM
SCHEMBL4749262 0.92 TP53 (0.75) TP53CREBBPKDM4EALDH1A1PKM
SCHEMBL31307876 0.89 TP53 (1.00) TP53CREBBPKDM4EALDH1A1PKM
SCHEMBL23493740 0.89 TP53 (1.00) TP53CREBBPKDM4EALDH1A1PKM
SCHEMBL5329104 0.86 CREBBP (0.82) TP53CREBBPKDM4EALDH1A1PKM
SCHEMBL5322774 0.86 CREBBP (0.82) TP53CREBBPKDM4EALDH1A1PKM
SCHEMBL5328005 0.86 PAX8 (0.83) TP53CREBBPKDM4EALDH1A1PKM
SCHEMBL5325640 0.85 PAX8 (0.85) TP53CREBBPKDM4EALDH1A1PKM
SCHEMBL31307791 0.84 TP53 (0.88) TP53CREBBPKDM4EALDH1A1PKM
SCHEMBL23494146 0.84 TP53 (0.88) TP53CREBBPKDM4EALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007139496-A1 QUINOLINE DERIVATIVES ACTING AS TYROSINE KINASE INHIBITORS CLANOTECH AB (SE) 2007-12-06 WO disclosed