SCHEMBL5326115

SCHEMBL5326115

Cc1ccc2c(c1)NC(=O)N(C1COc3ccccc3OC1)N=C2C1CCCCC1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTH1R Q03431 8/20 0.51
CYP19A1 P11511 2/20 0.36
HSD17B10 Q99714 3/20 0.35
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
CCKBR P32239 3/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5332531 0.91 PTH1R (0.44) PTH1RCYP19A1HSD17B10KDM4EALDH1A1
SCHEMBL5285662 0.86 CES2 (0.42) PTH1RHSD17B10KDM4EALDH1A1
SCHEMBL5322785 0.86 CES2 (0.42) PTH1RHSD17B10KDM4EALDH1A1
SCHEMBL5331038 0.86 CES2 (0.42) PTH1RHSD17B10KDM4EALDH1A1
SCHEMBL5326307 0.83 PTH1R (0.49) PTH1RHSD17B10KDM4EALDH1A1
SCHEMBL5330298 0.82 PTH1R (0.39) PTH1RHSD17B10KDM4EALDH1A1
SCHEMBL5319651 0.82 PTH1R (0.37) PTH1RHSD17B10KDM4EALDH1A1
SCHEMBL5320857 0.81 PTH1R (0.36) PTH1RHSD17B10KDM4EALDH1A1
SCHEMBL5281832 0.78 L3MBTL3 (0.42) KDM4EALDH1A1
SCHEMBL5323429 0.77 CES2 (0.42) PTH1RHSD17B10KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129120-A9 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2007-03-22 WO disclosed
WO-2006129120-A2 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2006-12-07 WO disclosed