SCHEMBL5327308

SCHEMBL5327308

CSc1ccc(-n2c(-c3ccc(C)cc3)cc(=O)n(CC(N)=NO)c2=O)cc1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
PTGS2 P35354 7/20 0.35
CHRNA7 P36544 1/20 0.34
SMN1; SMN2 Q16637 3/20 0.33
PTGS1 P23219 2/20 0.33
THRB P10828 1/20 0.33
CYP2C9 P11712 1/20 0.33
LMNA P02545 1/20 0.32
CYP2C19 P33261 1/20 0.32
TP53 P04637 1/20 0.32
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5325002 0.88 PTGS2 (0.35) HTTPTGS2CHRNA7SMN1; SMN2PTGS1
SCHEMBL5324999 0.88 PTGS2 (0.35) HTTPTGS2CHRNA7SMN1; SMN2PTGS1
SCHEMBL5288972 0.88 MEN1 (0.40) HTTMEN1KMT2ATDP1PTGS2
SCHEMBL5297375 0.85 MEN1 (0.42) HTTMEN1KMT2APTGS2CHRNA7
SCHEMBL5326545 0.85 PTGS2 (0.39) HTTMEN1KMT2APTGS2CHRNA7
SCHEMBL5331474 0.83 PTGS2 (0.38) HTTMEN1KMT2APTGS2CHRNA7
SCHEMBL14624165 0.82 LMNA (0.37) HTTNPC1RAB9APTGS2SMN1; SMN2
SCHEMBL5325697 0.82 RAD51 (0.40) HTTNPC1RAB9APTGS2CHRNA7
SCHEMBL14622895 0.82 PTGS2 (0.41) KMT2ATDP1PTGS2SMN1; SMN2CYP2C19
SCHEMBL5331619 0.82 PTGS2 (0.34) HTTKMT2ATDP1PTGS2CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007007161-A2 NOVEL BIO-ACTIVE DERIVATIVES ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-01-18 WO disclosed