SCHEMBL5327469

SCHEMBL5327469

COC(=O)C1=C(C)NC(=O)NC1c1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.71
TDP1 Q9NUW8 1/20 0.68
PKM P14618 1/20 0.67
GUSB P08236 1/20 0.67
ADORA2B P29275 1/20 0.64
KMT2A Q03164 2/20 0.63
POLB P06746 1/20 0.62
KDM4E B2RXH2 1/20 0.62
MEN1 O00255 1/20 0.62
ALDH1A1 P00352 1/20 0.62
THRB P10828 1/20 0.62
HSD17B10 Q99714 1/20 0.62
RAB9A P51151 1/20 0.61
TSHR P16473 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19752674 1.00 USP2 (0.71) USP2TDP1PKMGUSBADORA2B
SCHEMBL10279640 0.88 PKM (0.67) PKMGUSBADORA2BKMT2AKDM4E
SCHEMBL10112947 0.87 HSD17B10 (0.69) PKMGUSBADORA2BKMT2AKDM4E
SCHEMBL5347891 0.86 KIF11 (0.75) ADORA2BPOLBHSD17B10TSHR
SCHEMBL19752667 0.86 KIF11 (0.75) ADORA2BPOLBHSD17B10TSHR
SCHEMBL18025267 0.86 KIF11 (0.75) ADORA2BPOLBHSD17B10TSHR
SCHEMBL28595517 0.86 ALDH1A1 (0.78) PKMGUSBKMT2AKDM4EMEN1
SCHEMBL19732955 0.84 USP2 (0.79) USP2TDP1KMT2APOLBKDM4E
SCHEMBL13789190 0.84 USP2 (0.79) USP2TDP1KMT2APOLBKDM4E
SCHEMBL19732923 0.84 USP2 (0.79) USP2TDP1KMT2APOLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110437100-B Preparation method and application of novel ionic salicylaldehyde Schiff base zirconium complex 山西医科大学 2022-03-11 CN disclosed
WO-2007105233-A2 AN IMPROVED PROCESS FOR THE PREPARATION OF 4,5,6-SUBSTITUTED 3,4-DIHYDROPYRIMIDIN-2-ONES AND THEIR 2-THIOXO ANALOGUES COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2007-09-20 WO disclosed
US-5786472-A CATALYTIC CONDENSATION OF UREA WITH DIKETONES USIN BORON REAGENT AND ACID CATALYST MERCK & CO., INC. (US) 1998-07-28 US disclosed