SCHEMBL5328017

SCHEMBL5328017

CNC(=O)CCc1nccn1C(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
ACSS2 Q9NR19 1/20 0.40
NR4A2 P43354 1/20 0.38
HDAC6 Q9UBN7 2/20 0.38
EGFR P00533 1/20 0.36
SRC P12931 1/20 0.36
LMNA P02545 1/20 0.36
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35
NPC1 O15118 1/20 0.34
TP53 P04637 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5319750 0.85 MEN1 (0.41) KMT2AMEN1HDAC6LMNAMAPT
SCHEMBL7971128 0.85 ALDH1A1 (0.43) KMT2AMEN1EGFRSRCLMNA
SCHEMBL5325316 0.80 SMN1; SMN2 (0.43) KMT2AMEN1LMNATP53MAPT
SCHEMBL5320461 0.78 BLM (0.38) KMT2AMEN1NPC1
SCHEMBL1528022 0.78 KMT2A (0.44) KMT2AMEN1EGFRLMNATP53
SCHEMBL8806580 0.78 KMT2A (0.44) KMT2AMEN1LMNAMAPT
SCHEMBL6446028 0.76 KMT2A (0.43) KMT2AMEN1CYP1A2CYP2C19MAPT
SCHEMBL8806973 0.75 KMT2A (0.42) KMT2AMEN1
SCHEMBL4759513 0.75 KMT2A (0.42) KMT2AMEN1MAPT
SCHEMBL27544681 0.75 KMT2A (0.41) KMT2AMEN1EGFRLMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129120-A9 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2007-03-22 WO disclosed
WO-2006129120-A2 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2006-12-07 WO disclosed