SCHEMBL7971128

SCHEMBL7971128

COC(=O)CCc1nccn1C(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
RAB9A P51151 1/20 0.43
TSHR P16473 1/20 0.41
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
KDM4E B2RXH2 3/20 0.39
SMN1; SMN2 Q16637 2/20 0.37
EGFR P00533 1/20 0.36
SRC P12931 1/20 0.36
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
HSP90B1 P14625 1/20 0.36
CA12 O43570 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5325316 0.88 SMN1; SMN2 (0.43) ALDH1A1MEN1KMT2ARAB9AKDM4E
SCHEMBL5319750 0.85 MEN1 (0.41) ALDH1A1MEN1KMT2ASMN1; SMN2BLM
SCHEMBL5328017 0.85 KMT2A (0.40) MEN1KMT2AEGFRSRCLMNA
SCHEMBL5320461 0.83 BLM (0.38) ALDH1A1MEN1KMT2ARAB9AHSP90AA1
SCHEMBL1528022 0.78 KMT2A (0.44) MEN1KMT2ARAB9ATSHRCYP11B1
SCHEMBL8806580 0.78 KMT2A (0.44) ALDH1A1MEN1KMT2ACYP11B1CYP11B2
SCHEMBL8170659 0.77 TBXAS1 (0.41) ALDH1A1MEN1KMT2ATSHRSMN1; SMN2
SCHEMBL584666 0.76 KMT2A (0.43) MEN1KMT2ARAB9ATSHRCYP11B1
SCHEMBL6446028 0.76 KMT2A (0.43) MEN1KMT2ACYP11B1CYP11B2KDM4E
SCHEMBL8806973 0.75 KMT2A (0.42) ALDH1A1MEN1KMT2ACYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6316436-B1 ANTICANCER AGENTS MERCK & CO., INC. 2001-11-13 US disclosed