SCHEMBL5328503

SCHEMBL5328503

Cc1nc2c(O)c(CCC(=O)c3ccccc3)c(C(=O)NC3CC3)cn2c1C

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
KMT2A Q03164 1/20 0.38
BRD4 O60885 1/20 0.36
HPGDS O60760 2/20 0.36
RAB9A P51151 2/20 0.36
SMYD3 Q9H7B4 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
TP53 P04637 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
PANK1 Q8TE04 1/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5329533 0.87 CYP3A4 (0.36) KMT2ABRD4RAB9ATP53CYP3A4
SCHEMBL5327618 0.85 GLA (0.38) KMT2ARAB9ACYP3A4CYP2D6CYP2C9
Bicarbonate SCHEMBL5984921 0.84 GLA (0.37) KMT2ARAB9ACYP3A4CYP2D6CYP2C9
SCHEMBL5327517 0.83 MCHR1 (0.41) BRD4RAB9ANPC1
SCHEMBL5449403 0.83 MCHR1 (0.41) BRD4RAB9ANPC1
SCHEMBL5327514 0.83 MCHR1 (0.41) BRD4RAB9ANPC1
SCHEMBL5559185 0.82 KMT2A (0.42) ADRA1AKMT2ARAB9ATP53
SCHEMBL4994479 0.81 KMT2A (0.36) KMT2ARAB9ACYP3A4CYP2D6CYP2C9
SCHEMBL5330704 0.81 SMN1; SMN2 (0.43) KMT2ARAB9ATP53CYP2C9NPC1
Bicarbonate SCHEMBL4976269 0.81 KMT2A (0.35) KMT2ARAB9ACYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007141253-A1 PROCESS FOR THE PRODUCTION OF INTERMEDIATES FOR THE PREPARATION OF TRICYCLIC IMIDAZOPYRIDINES NYCOMED GMBH (DE) 2007-12-13 WO disclosed