SCHEMBL5329140

SCHEMBL5329140

CC(C)(C)OC(=O)N(N)[C@H]1CC[C@@](C#N)(c2ccccc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 5/20 0.50
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
CYP2D6 P10635 1/20 0.39
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
F11 P03951 2/20 0.38
CHRM4 P08173 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
OPRD1 P41143 1/20 0.37
GRM2 Q14416 1/20 0.36
PDE4B Q07343 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8063001 0.82 HSD11B1 (0.52) HSD11B1MEN1KMT2ACYP2D6F11
SCHEMBL13688478 0.79 HSD11B1 (0.47) HSD11B1MEN1KMT2ACA12CA1
SCHEMBL8052851 0.78 CHRM4 (0.55) HSD11B1MEN1KMT2ACHRM4
SCHEMBL8024304 0.76 KMT2A (0.52) HSD11B1MEN1KMT2ACYP2D6NPC1
SCHEMBL8101516 0.74 MEN1 (0.58) HSD11B1MEN1KMT2ACYP2D6NPC1
SCHEMBL5278104 0.74 HSD11B1 (0.44) HSD11B1NPC1RAB9A
SCHEMBL5286055 0.73 NPY5R (0.41)
SCHEMBL2529921 0.72 CA12 (0.54) CA12CA1CA2CA7CA9
SCHEMBL4367475 0.72 CHRM2 (0.34) HSD11B1
SCHEMBL28320948 0.70 OPRD1 (0.50) MEN1KMT2ACA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129120-A9 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2007-03-22 WO disclosed
WO-2006129120-A2 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2006-12-07 WO disclosed