SCHEMBL532978

SCHEMBL532978

Cc1cc(C)c(N2CCCC2)c(C)c1NS(=O)(=O)/C=C/c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.45
TSHR P16473 2/20 0.45
ALOX15 P16050 1/20 0.45
LMNA P02545 3/20 0.41
HTT P42858 2/20 0.41
KMT2A Q03164 3/20 0.40
POLB P06746 2/20 0.40
PKM P14618 1/20 0.40
HSP90AA1 P07900 2/20 0.40
MAPK1 P28482 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
GAA P10253 2/20 0.39
PTGES2 Q9H7Z7 1/20 0.39
GHSR Q92847 1/20 0.39
KDM4E B2RXH2 1/20 0.38
MEN1 O00255 1/20 0.38
HSD17B10 Q99714 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL532979 1.00 ALDH1A1 (0.45) ALDH1A1TSHRALOX15LMNAHTT
SCHEMBL532776 0.80 FFAR4 (0.54) ALDH1A1TSHRALOX15LMNAKMT2A
SCHEMBL533164 0.77 PTGES2 (0.39) LMNAKMT2APOLBPTGES2MEN1
SCHEMBL532980 0.77 JAK2 (0.48) ALDH1A1TSHRLMNAHTTKMT2A
SCHEMBL532988 0.76 ALDH1A1 (0.42) ALDH1A1TSHRKMT2APOLBMAPK1
SCHEMBL534077 0.76 TSHR (0.47) ALDH1A1TSHRLMNAKMT2APOLB
SCHEMBL533083 0.74 EDNRA (0.46) ALDH1A1LMNAPOLBSMN1; SMN2
SCHEMBL10092379 0.74 ALDH1A1 (0.31) ALDH1A1HTTPOLBSMN1; SMN2
SCHEMBL532038 0.74 ALDH1A1 (0.54) ALDH1A1TSHRLMNAKMT2APOLB
SCHEMBL532939 0.74 EDNRA (0.43) ALDH1A1KMT2APOLBGAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2415760-A2 CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2012-02-08 EP disclosed
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed
US-7319111-B2 Phenylenediamine Urotensin-II receptor antagonists and CCR-9 antagonists ENCYSIVE PHARMACEUTICALS, INC. (US) 2008-01-15 US disclosed